SCHEMBL8595148

SCHEMBL8595148

O=C(O)c1conc1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
KDM4E B2RXH2 6/20 0.39
MAPT P10636 3/20 0.39
ALOX15 P16050 2/20 0.39
TSHR P16473 2/20 0.39
CYP3A4 P08684 1/20 0.39
BLM P54132 1/20 0.39
AGER Q15109 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PTGS2 P35354 3/20 0.36
ASPH Q12797 1/20 0.36
KDM8 Q8N371 1/20 0.36
LDHA P00338 1/20 0.35
CYP1A2 P05177 1/20 0.35
HPGD P15428 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9567818 0.85 PTGS2 (0.34) ALDH1A1KDM4EMAPTALOX15TSHR
SCHEMBL9278686 0.85 IKBKB (0.36) ALDH1A1KDM4EMAPTALOX15TSHR
SCHEMBL8463065 0.78 PTGS2 (0.56) ALDH1A1KDM4EMAPTTSHRNPSR1
SCHEMBL353410 0.76
SCHEMBL4327521 0.76
SCHEMBL161729 0.76
SCHEMBL933947 0.76 ALDH1A1 (0.41) ALDH1A1KDM4EMAPTTSHRHPGD
SCHEMBL8957137 0.76 KDM4E (0.46) ALDH1A1KDM4EMAPTALOX15TSHR
SCHEMBL2696901 0.76 ALDH1A1 (0.44) ALDH1A1KDM4EMAPTTSHRL3MBTL1
SCHEMBL27654721 0.74 PTGS2 (0.43) ALDH1A1KDM4EMAPTPTGS2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0562382-B1 Process for the preparation of isoxazole-3,4-dicarboxylic acid derivatives BASF AG (DE) 1998-01-21 EP claimed
EP-0562377-B1 Preparation of isoxazole-3-carboxamide-4-carboxylic acid esters by selective amidation BASF AG (DE) 1997-05-14 EP claimed
US-5276160-A Amidation of primary or secondary amines BASF AKTIENGESELLSCHAFT (DE) 1994-01-04 US claimed
US-5264580-A Reaction of hydroximyl chlorides and beta-keto acids or esters, cyclization BASF AKTIENGESELLSCHAFT (DE) 1993-11-23 US claimed
JP-6016650-A None JP disclosed
CN-115232085-B Malonate compound, preparation method and application thereof 贵州工业职业技术学院 2023-09-05 CN disclosed
CN-115232085-A Malonate type compound, preparation method and application thereof 贵州理工学院 2022-10-25 CN disclosed
CN-105875625-A Method for producing novel rimsulfuron formulations and use thereof 龙灯农业化工国际有限公司 2016-08-24 CN disclosed
EP-0562382-B1 Process for the preparation of isoxazole-3,4-dicarboxylic acid derivatives BASF AG (DE) 1998-01-21 EP disclosed
US-5576270-A HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1996-11-19 US disclosed
JP-H0616650-A PRODUCTION OF 3-CARBAMOYLISOXAZOLE-4-CARBOXYLIC ESTER BASF AG 1994-01-25 JP disclosed
US-5276160-A Amidation of primary or secondary amines BASF AKTIENGESELLSCHAFT (DE) 1994-01-04 US disclosed
US-4137237-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1979-01-30 US disclosed
US-4093622-A Pyridine esters of cyclopropane-carboxylic acid ZOECON CORPORATION (US) 1978-06-06 US disclosed
US-4070475-A THIOALKYL-, AMINOALKYL-, AND OXYALKYL- SUBSTITUTED GUANIDINES SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1978-01-24 US disclosed
US-4024271-A INHIBITORS OF HISTAMINE ACTIVITY SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1977-05-17 US disclosed
US-4022797-A PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1977-05-10 US disclosed
US-4018931-A INHIBITION OF H-2 HISTAMINE RECEPTORS SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1977-04-19 US disclosed
US-3950333-A HISTAMINE INHIBITORS, OXYALKYL, THIOALKYL, AMINOALKYL DERIVATIVES SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1976-04-13 US disclosed
US-3950353-A HISTAMINE INHIBITORS SMITH KLINE & FRENCH LABORATORIES LIMITED (EN) 1976-04-13 US disclosed