SCHEMBL9282153

SCHEMBL9282153

CCOC(=O)CCc1ccc(C#Cc2cc3c(cc2CC)SC(C)(C)CC3(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.40
CYP4A11 Q02928 1/20 0.40
FFAR1 O14842 15/20 0.40
CHRM2 P08172 1/20 0.36
S1PR1 P21453 1/20 0.36
FPR1 P21462 1/20 0.36
FPR3 P25089 1/20 0.36
GPR183 P32249 1/20 0.36
APLNR P35414 1/20 0.36
FFAR4 Q5NUL3 1/20 0.36
GPR65 Q8IYL9 1/20 0.36
FDFT1 P37268 1/20 0.35
CYP4Z1 Q86W10 1/20 0.35
CYP3A4 P08684 1/20 0.35
RARA P10276 1/20 0.35
RARB P10826 1/20 0.35
RARG P13631 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700768 0.88 FFAR1 (0.53) FFAR1CHRM2S1PR1FPR1FPR3
SCHEMBL8876609 0.87 CYP3A4 (0.41) CYP4F2CYP4A11FFAR1FFAR4FDFT1
SCHEMBL9180592 0.84 RARA (0.46) CYP3A4RARARARBRARGKMT2A
SCHEMBL8865668 0.81 CYP3A4 (0.36) CYP4F2CYP4A11CYP3A4RARARARB
SCHEMBL8875500 0.81 CYP3A4 (0.40) CYP4F2CYP4A11FFAR1FFAR4CYP4Z1
SCHEMBL9176529 0.80 RARA (0.44) CYP3A4RARARARBRARGKMT2A
SCHEMBL9284407 0.80 RARA (0.35) CYP4F2CYP4A11FFAR1CYP3A4RARA
SCHEMBL8865478 0.79 CYP4F2 (0.34) CYP4F2CYP4A11FFAR1RARARARB
SCHEMBL8875274 0.79 CYP3A4 (0.41) CYP4F2CYP4A11FFAR1FFAR4FDFT1
SCHEMBL8865711 0.79 RARA (0.38) CYP3A4RARARARBRARGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0419131-B1 Acetylenes disubstituted with a phenyl group and a 2-substituted chromanyl, thiochromanyl or 1,2,3,4-tetrahydroquinolinyl group having retinoid-like activity ALLERGAN INC (US) 1995-07-05 EP disclosed
US-5278318-A Acetylation under Friedel Crafts condition ALLERGAN, INC. (US) 1994-01-11 US disclosed
US-4980369-A ANTIARTHRITIC AGENTS, SKIN DISORDERS, ANTIULCER AGENTS, WOUND HEALING AGENTS ALLERGAN, INC. (US) 1990-12-25 US disclosed