SCHEMBL9284693

SCHEMBL9284693

COc1[nH]nc(-c2ccc(Br)cc2)c1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.44
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
IKBKB O14920 1/20 0.40
CHUK O15111 1/20 0.40
DCLK1 O15075 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
CHEK2 O96017 1/20 0.39
CSF1R P07333 1/20 0.39
FER P16591 1/20 0.39
CDK2 P24941 1/20 0.39
MARK3 P27448 1/20 0.39
FLT4 P35916 1/20 0.39
FLT3 P36888 1/20 0.39
MAPK9 P45984 1/20 0.39
CSNK1D P48730 1/20 0.39
CLK2 P49760 1/20 0.39
CSNK2A1 P68400 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10922767 0.81 MKNK1 (0.41) RAB9ASMN1; SMN2CDK2DYRK1AMEN1
Hydrochloric Acid SCHEMBL10987600 0.79 MKNK1 (0.41) RAB9ASMN1; SMN2CDK2DYRK1AMEN1
SCHEMBL9182327 0.76 IKBKB (0.47) CHEK1NPC1RAB9ASMN1; SMN2IKBKB
SCHEMBL9183883 0.75 CNR1 (0.47) CHEK1NPC1RAB9ASMN1; SMN2IKBKB
SCHEMBL27759841 0.75 CDK2 (0.45) CHEK1NPC1RAB9ASMN1; SMN2DCLK1
SCHEMBL11070855 0.73 RAB9A (0.50) RAB9ASMN1; SMN2MEN1KMT2ATP53
SCHEMBL10981820 0.72 MAP2K4 (0.52) CHEK1NPC1SMN1; SMN2PRKD3MAP4K4
SCHEMBL2614356 0.68 IKBKB (0.50) CHEK1NPC1RAB9ASMN1; SMN2IKBKB
SCHEMBL14712058 0.67 HSP90AA1 (0.56) NPC1RAB9ASMN1; SMN2IKBKBCHUK
SCHEMBL15741508 0.67 NPC1 (0.43) CHEK1NPC1RAB9ASMN1; SMN2IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656897-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LIMITED (GB) 1995-06-14 EP disclosed
WO-1994005660-A1 QUINUCLIDINE DERIVATIVES AS SQUALENE SYNTHASE INHIBITORS ZENECA LIMITED (GB) 1994-03-17 WO disclosed