SCHEMBL15741508

SCHEMBL15741508

Cc1c[nH]nc1-c1ccc(Br)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
IKBKB O14920 1/20 0.41
CHUK O15111 1/20 0.41
ERBB2 P04626 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
METAP2 P50579 1/20 0.37
ATM Q13315 1/20 0.37
ALDH1A1 P00352 2/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
GPR55 Q9Y2T6 1/20 0.36
PTGS2 P35354 1/20 0.36
CHEK1 O14757 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
USP2 O75604 1/20 0.35
MAPK13 O15264 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6850964 0.83 MEN1 (0.48) SMN1; SMN2ERBB2KDM4EMAPTMETAP2
SCHEMBL3755589 0.80 IKBKB (0.41) IKBKBERBB2KDM4EMETAP2
SCHEMBL3160320 0.80 MAPK14 (0.42) NPC1RAB9ASMN1; SMN2ERBB2KDM4E
SCHEMBL13363877 0.80 ERBB2 (0.39) NPC1RAB9ASMN1; SMN2ERBB2MAPT
SCHEMBL2449809 0.79 ALOX15 (0.48) NPC1RAB9ASMN1; SMN2KDM4EMAPT
SCHEMBL5223142 0.78 MEN1 (0.53) NPC1RAB9AKDM4EMAPTALDH1A1
SCHEMBL15186271 0.78 LMNA (0.40) MAPTALDH1A1MAPK13MAPK12MAPK11
Hydrochloric Acid SCHEMBL30879670 0.77 MEN1 (0.51) NPC1RAB9AKDM4EMAPTALDH1A1
SCHEMBL14572024 0.77 ERBB2 (0.46) NPC1RAB9ASMN1; SMN2ERBB2KDM4E
SCHEMBL8806952 0.76 MAP2K4 (0.49) IKBKBCHUKCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922842-A2 NOVEL INHIBITOR COMPOUNDS OF PHOSPHODIESTERASE TYPE 10A AbbVie Inc. (US) 2015-09-30 EP disclosed
WO-2014079995-A2 NOVEL INHIBITOR COMPOUNDS OF PHOSPHODIESTERASE TYPE 10A ABBVIE INC. (US) 2014-05-30 WO disclosed