SCHEMBL9285136

SCHEMBL9285136

O=C(O)c1ccc(NS(=O)(=O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 1/20 0.74
CES1 P23141 1/20 0.73
CA12 O43570 1/20 0.71
CA1 P00915 1/20 0.71
CA2 P00918 1/20 0.71
CA9 Q16790 1/20 0.71
KMT2A Q03164 3/20 0.67
MEN1 O00255 2/20 0.67
MAPK1 P28482 1/20 0.64
HDAC3 O15379 1/20 0.62
HDAC4 P56524 1/20 0.62
HDAC1 Q13547 1/20 0.62
HDAC7 Q8WUI4 1/20 0.62
HDAC2 Q92769 1/20 0.62
HDAC10 Q969S8 1/20 0.62
HDAC11 Q96DB2 1/20 0.62
HDAC8 Q9BY41 1/20 0.62
HDAC6 Q9UBN7 1/20 0.62
HDAC9 Q9UKV0 1/20 0.62
HDAC5 Q9UQL6 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13028457 0.95 WDR5 (0.68) WDR5CES1CA12CA1CA2
SCHEMBL3558356 0.91 WDR5 (0.63) WDR5CES1CA12CA1CA2
SCHEMBL6554630 0.86 CES1 (1.00) WDR5CES1KMT2AMEN1HDAC1
SCHEMBL2474197 0.86 CES1 (1.00) WDR5CES1KMT2AMEN1HDAC1
SCHEMBL28262522 0.85 MAPT (0.74) WDR5CES1CA12CA9KMT2A
SCHEMBL7932062 0.85 CA12 (0.73) CA12CA1CA2CA9KMT2A
SCHEMBL893905 0.84 CA12 (0.73) CA12CA1CA2CA9KMT2A
SCHEMBL3715141 0.84 CA12 (0.75) CA12CA1CA2CA9KMT2A
SCHEMBL11047587 0.84 MEN1 (0.76) WDR5CES1CA12CA9KMT2A
SCHEMBL1834055 0.83 CA12 (0.71) WDR5CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102395270-B Novel compounds, pharmaceutical compositions containing same, methods of use for same, and methods for preparing same FASGEN INC 2014-11-12 CN disclosed
CN-102395270-A Novel compounds, pharmaceutical compositions containing same, methods of use for same, and methods for preparing same FASGEN INC 2012-03-28 CN disclosed
WO-1995004740-A1 7α-AMINO-1,1-DIOXOCEFEM L-VALYLAMIDES DOMPE' S.P.A. (IT) 1995-02-16 WO disclosed