SCHEMBL9285608

SCHEMBL9285608

CC(=O)Nc1ncc(-c2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)s1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.51
GAA P10253 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
PTGS1 P23219 7/20 0.46
PTGS2 P35354 5/20 0.46
CCNE2 O96020 5/20 0.43
CCNE1 P24864 5/20 0.43
CDK2 P24941 5/20 0.43
PIK3CG P48736 3/20 0.42
PIK3CD O00329 1/20 0.42
PIK3R1 P27986 1/20 0.42
PIK3CA P42336 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
KDR P35968 1/20 0.42
CCNB2 O95067 2/20 0.41
CDK1 P06493 2/20 0.41
CDK4 P11802 2/20 0.41
CCNB1 P14635 2/20 0.41
CCND1 P24385 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9179011 0.79 PTGS1 (0.68) ALDH1A1GAATDP1PTGS1PTGS2
SCHEMBL7127478 0.74 PTGS1 (0.58) PTGS1PTGS2CA1CA2
SCHEMBL5840422 0.74 KDR (0.72) CCNE2CCNE1CDK2KDRLIMK1
SCHEMBL17632040 0.71 ABL1 (0.62) CCNE2CCNE1CDK2PIK3CGKDR
SCHEMBL179490 0.71 CCNE1 (0.52) CCNE2CCNE1CDK2PIK3CGPIK3CA
SCHEMBL3901196 0.71 ATAD2 (0.45) CCNE1CDK2PIK3CGPIK3CDPIK3R1
SCHEMBL6916158 0.71 ERCC1 (0.53) CCNE2CCNE1CDK2PIK3CGPIK3CD
SCHEMBL12991170 0.71 MEN1 (0.48) CCNE2CCNE1CDK2PIK3CGPIK3CD
SCHEMBL4307403 0.70 LIMK1 (0.51) CCNE2CCNE1CDK2PIK3CGPIK3CA
SCHEMBL12496031 0.69 KDR (0.50) CCNE2CCNE1CDK2PIK3CAKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0371438-B1 3,5-Di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxiphenyl- 1,2,4-thiadiazoles, -oxadiazoles as antiinflammatory agents WARNER LAMBERT CO (US) 1995-08-30 EP disclosed
US-5155122-A Cyclooxygenase, lipoxygenase inhibitors WARNER-LAMBERT COMPANY (US) 1992-10-13 US disclosed