SCHEMBL9287384

SCHEMBL9287384

CCCN(Cc1cccnc1)c1ccccc1C

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.50
CHRNA4 P43681 2/20 0.50
HTT P42858 1/20 0.43
CYP3A4 P08684 1/20 0.43
GRM2 Q14416 5/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CHRNA7 P36544 1/20 0.43
NR1H2 P55055 1/20 0.41
NR1H3 Q13133 1/20 0.41
NAMPT P43490 1/20 0.41
NOTUM Q6P988 1/20 0.40
RIPK1 Q13546 1/20 0.40
KCNN4 O15554 1/20 0.40
KCNA5 P22460 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9288516 0.85 KCNA5 (0.40) CHRNB2CHRNA4KCNA5
SCHEMBL9288362 0.84 CYP3A4 (0.54) CHRNB2CHRNA4CYP3A4GRM2TDP1
SCHEMBL6584770 0.81 CHRNB2 (0.54) CHRNB2CHRNA4GRM2NR1H2NR1H3
SCHEMBL9284721 0.79 CYP3A4 (0.41) CYP3A4TDP1NOTUMKCNN4KCNA5
SCHEMBL10980698 0.78 CYP3A4 (0.45) CHRNB2CHRNA4HTTCYP3A4GRM2
SCHEMBL9284419 0.77 CYP3A4 (0.52) CHRNB2CHRNA4CYP3A4GRM2TDP1
SCHEMBL10995093 0.77 S1PR1 (0.47) CHRNB2CHRNA4HTTCYP3A4GRM2
SCHEMBL516401 0.76 CRHR1 (0.44) CYP3A4
SCHEMBL12653608 0.74 NR1H2 (0.48) NR1H2NR1H3
Hydrochloric Acid SCHEMBL11023677 0.74 CRHR1 (0.43) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012075232-A1 OPIOID RECEPTOR LIGANDS AND METHODS OF USING AND MAKING THE SAME TREVENA, INC. (US) 2012-06-07 WO disclosed