SCHEMBL9290707

SCHEMBL9290707

C=CCc1cnc(N)nc1C

nearest known ligand 0.51

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.47
SLC2A1 P11166 1/20 0.39
PDXK O00764 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9102557 0.78 DHFR (0.44) DHFR
SCHEMBL9607552 0.76 DHFR (0.51) DHFR
Guanidine SCHEMBL11341298 0.75 DHFR (0.53) DHFR
SCHEMBL5807751 0.75 DHFR (0.45) DHFRPDXK
SCHEMBL23094501 0.75 LMNA (0.50) PDXK
SCHEMBL14076717 0.75 DHFR (0.38) DHFR
Hydrochloric Acid SCHEMBL28160879 0.75 DHFR (0.50) DHFR
SCHEMBL28938199 0.74 NUDT1 (0.53) DHFR
SCHEMBL9286815 0.73 HSP90AA1 (0.47) DHFR
SCHEMBL27523630 0.73 DHFR (0.48) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012071501-A1 BENZOXAZEPINES ASN INHIBITORS OF P13K/M TOR AND METHODS OF THEIR USE AND MANUFACTURE EXELIXIS, INC. (US) 2012-05-31 WO disclosed