SCHEMBL9292425

SCHEMBL9292425

O=C(O)Cc1c([N+](=O)[O-])cc([N+](=O)[O-])cc1[N+](=O)[O-]

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.64
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
ALDH1A1 P00352 8/20 0.50
KMT2A Q03164 6/20 0.50
GPR35 Q9HC97 5/20 0.50
MEN1 O00255 5/20 0.50
MAPT P10636 4/20 0.50
MAPK1 P28482 4/20 0.50
TDP1 Q9NUW8 2/20 0.50
HPGD P15428 2/20 0.50
CYP2C9 P11712 2/20 0.50
KDM4E B2RXH2 1/20 0.50
TTR P02766 1/20 0.50
ALOX15 P16050 1/20 0.50
ALOX12 P18054 1/20 0.50
RECQL P46063 1/20 0.50
PMP22 Q01453 1/20 0.50
HIF1A Q16665 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2711927 0.88 GPR35 (0.57) CYP1A2CA1CA2ALDH1A1KMT2A
SCHEMBL2711921 0.88 GPR35 (0.57) CYP1A2CA1CA2ALDH1A1KMT2A
SCHEMBL10617906 0.88 ALDH1A1 (0.57) CYP1A2CA1CA2ALDH1A1KMT2A
SCHEMBL10619763 0.86 CYP1A2 (0.58) CYP1A2CA1CA2ALDH1A1KMT2A
SCHEMBL6445564 0.84 CYP1A2 (0.47) CYP1A2CA1CA2ALDH1A1KMT2A
SCHEMBL11797519 0.84 KMT2A (0.54) CYP1A2CA1CA2ALDH1A1KMT2A
SCHEMBL11797508 0.84 KMT2A (0.54) CYP1A2CA1CA2ALDH1A1KMT2A
SCHEMBL4319842 0.82 CYP1A2 (0.49) CYP1A2ALDH1A1KMT2AMEN1MAPT
(Z)-1,2-Diphenylethene SCHEMBL9766302 0.81 CYP1A2 (0.49) CYP1A2ALDH1A1KMT2AMEN1MAPT
SCHEMBL1407953 0.81 ALDH1A1 (0.53) CYP1A2CA1CA2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0491831-A4 1994-01-05 EP disclosed
EP-0491831-A1 PROCESS FOR THE PRODUCTION OF ESTERS EXHIBITING NONLINEAR OPTICAL RESPONSE HOECHST CELANESE CORPORATION (US) 1992-07-01 EP disclosed
WO-1991003683-A1 ACRYLIC COPOLYMERS EXHIBITING NONLINEAR OPTICAL RESPONSE HOECHST CELANESE CORP (US) 1991-03-21 WO disclosed
WO-1991003457-A1 PROCESS FOR THE PRODUCTION OF ESTERS EXHIBITING NONLINEAR OPTICAL RESPONSE HOECHST CELANESE CORPORATION (US) 1991-03-21 WO disclosed
US-4997977-A Process for the production of esters exhibiting nonlinear optical response HOECHST CELANESE CORP. (US) 1991-03-05 US disclosed