SCHEMBL9298985

SCHEMBL9298985

O=C(O)C1(c2ncc[nH]2)CCCc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC9 Q9UKV0 1/20 0.43
AKR1B1 P15121 1/20 0.41
KDM5A P29375 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
ALDH1A1 P00352 2/20 0.37
ADRA2A P08913 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
TSHR P16473 2/20 0.36
AKR1C1 Q04828 1/20 0.36
MEN1 O00255 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL779741 0.80 ADRA1A (0.39) AKR1B1ALDH1A1ADRA2AADRA1DADRA1A
SCHEMBL9531758 0.73 TSHR (0.40) HDAC9ALDH1A1ADRA2AADRA1DADRA1A
SCHEMBL4432306 0.70 HDAC9 (0.71) HDAC9TSHRAKR1C1KDM1A
SCHEMBL14214917 0.70 HDAC9 (0.57) HDAC9AKR1B1TSHRAKR1C1MEN1
SCHEMBL4851505 0.69 KDM1A (0.50) HDAC9AKR1B1KDM5AKDM4CKDM5B
SCHEMBL30219063 0.69 AKR1C1 (0.48) HDAC9AKR1B1TSHRAKR1C1MEN1
SCHEMBL687495 0.69 AKR1C1 (0.48) HDAC9AKR1B1TSHRAKR1C1MEN1
SCHEMBL28941603 0.68 HDAC9 (0.43) HDAC9AKR1B1TSHRAKR1C1CYP3A4
SCHEMBL27728415 0.68 HDAC9 (0.55) HDAC9KDM5AKDM4CKDM5BALDH1A1
SCHEMBL367096 0.67 AKR1C1 (0.47) HDAC9AKR1B1TSHRAKR1C1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354770-A Cardiovascular system disorders DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1994-10-11 US disclosed