Bucillamine

Bucillamine

SCHEMBL930021

CC(C)(S)C(=O)N[C@H](CS)C(=O)O

nearest known ligand 0.59

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.59
KDM4E B2RXH2 1/20 0.59
THRB P10828 1/20 0.59
ALOX15 P16050 1/20 0.59
NFKB1 P19838 1/20 0.59
PTGS2 P35354 1/20 0.59
THPO P40225 1/20 0.59
RECQL P46063 1/20 0.59
BLM P54132 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
ACE P12821 3/20 0.54
MME P08473 1/20 0.54
ACE2 Q9BYF1 1/20 0.54
FOLH1 Q04609 4/20 0.50
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
NAALAD2 Q9Y3Q0 3/20 0.35
RIMKLA Q8IXN7 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bucillamine SCHEMBL5060887 1.00 MAPT (0.59) MAPTKDM4ETHRBALOX15NFKB1
Bucillamine SCHEMBL522713 1.00 MAPT (0.59) MAPTKDM4ETHRBALOX15NFKB1
Bucillamine SCHEMBL121965 1.00 MAPT (0.59) MAPTKDM4ETHRBALOX15NFKB1
Bucillamine SCHEMBL4632094 0.91 MAPT (0.50) MAPTKDM4ETHRBALOX15NFKB1
Bucillamine SCHEMBL28086441 0.88 PTGS1 (0.56) MAPTKDM4ETHRBALOX15NFKB1
SCHEMBL6661780 0.86 KDM4E (0.61) MAPTKDM4ETHRBALOX15NFKB1
SCHEMBL6661779 0.86 KDM4E (0.61) MAPTKDM4ETHRBALOX15NFKB1
SCHEMBL9324856 0.86 KDM4E (0.61) MAPTKDM4ETHRBALOX15NFKB1
SCHEMBL929192 0.85 ACE (0.51) MAPTKDM4ETHRBALOX15NFKB1
SCHEMBL929188 0.85 ACE (0.51) MAPTKDM4ETHRBALOX15NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7875268-B2 The use of certain dimercaptoamides as reducing agents, 2-mercapto-N-(2-mercaptoethyl)acetamide, results in curling that is satisfactoryin terms of intensity and in terms of hold over time; less substantial degradation of the hair fiber compared with the reducing agents of the prior art; permanent waves L'OREAL S.A. (FR) 2011-01-25 US claimed
EP-1584615-B1 Use of dimercaptoamides for permanently deforming of keratinic fibres OREAL (FR) 2008-05-28 EP claimed
US-20060013784-A1 Novel dimercaptoamides, compositions comprising them as reducing agents, and processes for permanently reshaping keratin fibers therewith L'OREAL S.A. (FR) 2006-01-19 US claimed
EP-1584615-A1 Use of dimercaptoamides for permanently deforming of keratinic fibres L'OREAL (FR) 2005-10-12 EP claimed
US-20230181607-A1 THIOSACCHARIDES FOR USE IN TREATING CORONAVIRUS INFECTION The University of the Regents of California (US) 2023-06-15 US disclosed
US-20230181607-A1 THIOSACCHARIDES FOR USE IN TREATING CORONAVIRUS INFECTION The University of the Regents of California (US) 2023-06-15 US disclosed
US-20230172885-A1 THIOL-CONTAINING COMPOUNDS FOR USE IN TREATING CORONAVIRUS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-06-08 US disclosed
US-20230172885-A1 THIOL-CONTAINING COMPOUNDS FOR USE IN TREATING CORONAVIRUS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2023-06-08 US disclosed
WO-2021231421-A1 THIOL-CONTAINING COMPOUNDS FOR USE IN TREATING CORONAVIRUS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-18 WO disclosed
WO-2021231397-A1 THIOSACCHARIDES FOR USE IN TREATING CORONAVIRUS INFECTION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-18 WO disclosed
US-20210154161-A1 MODIFIED-RELEASE BUCILLAMINE COMPOSITIONS, KITS, AND METHODS FOR TREATING CYSTINURIA, ARTHRITIS, GOUT, AND RELATED DISORDERS ALTIBIO INC (US) 2021-05-27 US disclosed
EP-3658130-A1 MODIFIED-RELEASE BUCILLAMINE COMPOSITIONS, KITS, AND METHODS FOR TREATING CYSTINURIA, ARTHRITIS, GOUT, AND RELATED DISORDERS Altibio, Inc. (US) 2020-06-03 EP disclosed
WO-2019023346-A1 MODIFIED-RELEASE BUCILLAMINE COMPOSITIONS, KITS, AND METHODS FOR TREATING CYSTINURIA, ARTHRITIS, GOUT, AND RELATED DISORDERS ALTIBIO, INC. (US) 2019-01-31 WO disclosed
WO-2019023346-A1 MODIFIED-RELEASE BUCILLAMINE COMPOSITIONS, KITS, AND METHODS FOR TREATING CYSTINURIA, ARTHRITIS, GOUT, AND RELATED DISORDERS ALTIBIO, INC. (US) 2019-01-31 WO disclosed
US-7875268-B2 The use of certain dimercaptoamides as reducing agents, 2-mercapto-N-(2-mercaptoethyl)acetamide, results in curling that is satisfactoryin terms of intensity and in terms of hold over time; less substantial degradation of the hair fiber compared with the reducing agents of the prior art; permanent waves L'OREAL S.A. (FR) 2011-01-25 US disclosed
EP-1584615-B1 Use of dimercaptoamides for permanently deforming of keratinic fibres OREAL (FR) 2008-05-28 EP disclosed
US-20060013784-A1 Novel dimercaptoamides, compositions comprising them as reducing agents, and processes for permanently reshaping keratin fibers therewith L'OREAL S.A. (FR) 2006-01-19 US disclosed
EP-1584615-A1 Use of dimercaptoamides for permanently deforming of keratinic fibres L'OREAL (FR) 2005-10-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060013784-A1 Novel dimercaptoamides, compositions comprising them as reducing agents, and processes for permanently reshaping keratin fibers therewith KRT18, CKAP4, S100A4 MAPT 998/4885KDM4E 488/4885THRB 4302/4885
US-20230172885-A1 THIOL-CONTAINING COMPOUNDS FOR USE IN TREATING CORONAVIRUS CTH, SARS1, CBS MAPT 1085/4885KDM4E 3990/4885THRB 3581/4885
US-20210154161-A1 MODIFIED-RELEASE BUCILLAMINE COMPOSITIONS, KITS, AND METHODS FOR TREATING CYSTINURIA, ARTHRITIS, GOUT, AND RELATED DISORDERS SLC7A11, CBS, SSB MAPT 4256/4885KDM4E 4591/4885THRB 1122/4885
US-20230181607-A1 THIOSACCHARIDES FOR USE IN TREATING CORONAVIRUS INFECTION TMPRSS4, ACE, ACE2 MAPT 2951/4885KDM4E 4488/4885THRB 1674/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.