SCHEMBL9300759

SCHEMBL9300759

CC(Nc1cc(CO)cc(Nc2c3ccccc3nc3ccccc23)c1C(C)S(C)(=O)=O)S(C)(=O)=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2B Q02880 9/20 0.53
TOP2A P11388 8/20 0.53
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CASP1 P29466 2/20 0.41
CASP7 P55210 2/20 0.41
KDM1A O60341 2/20 0.41
GLA P06280 2/20 0.41
SLC22A1 O15245 1/20 0.41
ABCC4 O15439 1/20 0.41
NR1I2 O75469 1/20 0.41
TP53 P04637 1/20 0.41
CYP3A4 P08684 1/20 0.41
CHRM1 P11229 1/20 0.41
TOP1 P11387 1/20 0.41
DRD2 P14416 1/20 0.41
TSHR P16473 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9547241 0.78 TOP2A (0.51) TOP2BTOP2AKDM1AGLARAB9A
SCHEMBL9300528 0.74 ELANE (0.48) TOP2BTOP2AGLATSHROPRD1
SCHEMBL9300541 0.74 TOP2B (0.48) TOP2BTOP2ACYP1A2CYP2D6CYP2C9
SCHEMBL9547262 0.74 TOP2A (0.46) TOP2BTOP2AKDM1AGLAOPRD1
SCHEMBL9300661 0.71 TOP2A (0.47) TOP2BTOP2AKDM1AGLATSHR
SCHEMBL9300901 0.71 KDM4E (0.48) TOP2BTOP2AKDM1AGLATSHR
SCHEMBL9299716 0.71 POLB (0.43) TOP2BTOP2AGLAKMT2AMEN1
SCHEMBL9300764 0.70 TOP2B (0.53) TOP2BTOP2ACYP1A2CYP2D6CYP2C9
SCHEMBL9302146 0.70 TOP2A (1.00) TOP2BTOP2ACYP1A2CYP2D6CYP2C9
SCHEMBL9300635 0.69 KDM4E (0.42) TOP2BTOP2AGLARAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354864-A Antitumor agents SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-10-11 US claimed
WO-1993023049-A1 3-(9-ACRIDINYLAMINO)-5-HYDROXYMETHYLANILINE DERIVATIVES AS ANTICANCER AGENTS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1993-11-25 WO claimed
US-5354864-A Antitumor agents SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1994-10-11 US disclosed