SCHEMBL9301210

SCHEMBL9301210

COc1ccc2c(-c3ccccc3)cc(C(=O)O)cc2c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 1/20 0.68
KDM4E B2RXH2 5/20 0.58
ALDH1A1 P00352 4/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
HPGD P15428 2/20 0.51
KMT2A Q03164 4/20 0.48
MAPT P10636 3/20 0.48
MEN1 O00255 3/20 0.48
NPSR1 Q6W5P4 2/20 0.47
ACACA Q13085 1/20 0.47
ALOX5 P09917 1/20 0.47
PIN1 Q13526 1/20 0.47
LMNA P02545 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
CYP3A4 P08684 2/20 0.46
NPC1 O15118 1/20 0.46
TP53 P04637 1/20 0.46
RAB9A P51151 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9300510 0.81 P2RY14 (1.00) P2RY14KDM4EALDH1A1HPGDKMT2A
SCHEMBL29120670 0.81 BACE1 (0.62) P2RY14KDM4EALDH1A1SMN1; SMN2HPGD
SCHEMBL9301722 0.79 P2RY14 (0.63) P2RY14KDM4EALDH1A1HPGDKMT2A
SCHEMBL12193502 0.79 KDM4E (0.65) P2RY14KDM4EALDH1A1HPGDLMNA
SCHEMBL3924343 0.79 ALDH1A1 (0.57) KDM4EALDH1A1SMN1; SMN2HPGDKMT2A
SCHEMBL10988314 0.78 MEN1 (0.59) P2RY14KDM4EALDH1A1HPGDKMT2A
SCHEMBL27335273 0.75 GPR84 (0.52) KDM4EALDH1A1SMN1; SMN2HPGDMAPT
SCHEMBL9303054 0.75 P2RY14 (0.55) P2RY14CYP3A4
SCHEMBL6204953 0.75 P2RY14 (0.61) P2RY14KDM4ESMN1; SMN2KMT2AMEN1
SCHEMBL6735457 0.75 PDE4B (0.51) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1087907-A Heteroaryl naphthalene as white (cell) triolefin biosynthesis inhibitor MERCK FROSST CANADA INC (CA) 1994-06-15 CN disclosed
US-5308852-A Cardiovascular disorders MERCK FROSST CANADA, INC. (CA) 1994-05-03 US disclosed
EP-0579304-A1 Heteroarylnaphthalenes as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1994-01-19 EP disclosed
WO-1994000444-A1 HETEROARYLNAPHTHALENES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1994-01-06 WO disclosed