SCHEMBL9300510

SCHEMBL9300510

O=C(O)c1cc(-c2ccccc2)c2ccc(OCc3ccccc3)cc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 1/20 1.00
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
ALOX5 P09917 3/20 0.56
LTB4R Q15722 1/20 0.56
LTB4R2 Q9NPC1 1/20 0.56
MRGPRX4 Q96LA9 2/20 0.55
NR4A2 P43354 3/20 0.55
NR4A1 P22736 1/20 0.55
NR4A3 Q92570 1/20 0.55
MAOB P27338 1/20 0.54
KDM4E B2RXH2 1/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
HPGD P15428 1/20 0.53
SRD5A2 P31213 1/20 0.53
HSD17B10 Q99714 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301439 0.88 P2RY14 (0.78) P2RY14ALOX5LTB4RLTB4R2MRGPRX4
SCHEMBL9300644 0.88 P2RY14 (0.78) P2RY14ALOX5LTB4RLTB4R2MAOB
SCHEMBL9301058 0.85 P2RY14 (0.73) P2RY14ALOX5LTB4RLTB4R2MRGPRX4
SCHEMBL9301072 0.83 P2RY14 (0.71) P2RY14ALOX5LTB4RLTB4R2MAOB
SCHEMBL2933136 0.83 P2RY14 (0.70) P2RY14ALOX5LTB4RLTB4R2MRGPRX4
SCHEMBL9301210 0.81 P2RY14 (0.68) P2RY14MEN1KMT2AALOX5KDM4E
SCHEMBL5921632 0.81 MRGPRX4 (0.76) P2RY14MEN1KMT2AALOX5MRGPRX4
Hydrochloric Acid SCHEMBL8380168 0.79 MRGPRX4 (0.74) P2RY14MEN1KMT2AALOX5MRGPRX4
SCHEMBL9302530 0.79 P2RY14 (0.63) P2RY14ALOX5MRGPRX4
SCHEMBL2934240 0.79 P2RY14 (0.65) P2RY14ALOX5LTB4RLTB4R2MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5308852-A Cardiovascular disorders MERCK FROSST CANADA, INC. (CA) 1994-05-03 US disclosed
EP-0579304-A1 Heteroarylnaphthalenes as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1994-01-19 EP disclosed
WO-1994000444-A1 HETEROARYLNAPHTHALENES AS INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS MERCK FROSST CANADA INC. (CA) 1994-01-06 WO disclosed