SCHEMBL9301219

SCHEMBL9301219

C=C(c1cccc([N+](=O)[O-])c1)c1nccn1C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.46
ALDH1A1 P00352 5/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
L3MBTL1 Q9Y468 3/20 0.45
LMNA P02545 2/20 0.45
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TP53 P04637 1/20 0.40
TSHR P16473 2/20 0.40
KDM4E B2RXH2 2/20 0.39
ALOX5 P09917 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23213140 0.78 ALDH1A1 (0.48) MAPTALDH1A1SMN1; SMN2LMNANPC1
SCHEMBL29796135 0.78 ALDH1A1 (0.48) MAPTALDH1A1SMN1; SMN2LMNANPC1
SCHEMBL7101531 0.77 MAPT (0.46) MAPTALDH1A1SMN1; SMN2L3MBTL1LMNA
SCHEMBL9301216 0.76 MAPT (0.49) MAPTALDH1A1SMN1; SMN2L3MBTL1LMNA
SCHEMBL9301223 0.76 MAPT (0.49) MAPTALDH1A1SMN1; SMN2L3MBTL1LMNA
SCHEMBL9545603 0.73 ALDH1A1 (0.52) MAPTALDH1A1L3MBTL1MEN1KMT2A
SCHEMBL30822838 0.71 MAPT (0.62) MAPTALDH1A1SMN1; SMN2L3MBTL1LMNA
SCHEMBL4746148 0.71 MAPT (0.62) MAPTALDH1A1SMN1; SMN2L3MBTL1LMNA
SCHEMBL27449893 0.70 CES2 (0.59) MAPTALDH1A1SMN1; SMN2L3MBTL1LMNA
SCHEMBL4717161 0.70 HSP90AA1 (0.46) MAPTALDH1A1SMN1; SMN2LMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360802-A Antagonists of cholecystokinin and gastrin MERCK SHARPE & DOHME LTD. 1994-11-01 US disclosed
EP-0514133-A1 Benzodiazepine derivatives, compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1992-11-19 EP disclosed