SCHEMBL9301541

SCHEMBL9301541

CCS(=O)(=O)NC(=O)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.58
MEN1 O00255 4/20 0.58
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
CYP2C9 P11712 1/20 0.57
ALDH1A1 P00352 4/20 0.56
ATM Q13315 1/20 0.56
HPGD P15428 2/20 0.55
GAA P10253 2/20 0.55
LMNA P02545 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
CES2 O00748 1/20 0.55
CES1 P23141 1/20 0.55
THRA P10827 1/20 0.54
TP53 P04637 1/20 0.54
POLB P06746 1/20 0.54
MAPT P10636 1/20 0.54
BLM P54132 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.53
TSHR P16473 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6639356 0.85 KMT2A (0.61) KMT2AMEN1ALDH1A1ATMHPGD
SCHEMBL10769076 0.82 KMT2A (0.57) KMT2AMEN1ALDH1A1HPGDGAA
SCHEMBL8548910 0.82 KMT2A (0.57) KMT2AMEN1ALDH1A1ATMHPGD
SCHEMBL9301197 0.82 ALDH1A1 (0.57) KMT2AMEN1ALDH1A1HPGDGAA
SCHEMBL8884550 0.81 ATM (0.67) KMT2AMEN1CYP1A2CYP3A4CYP2C9
SCHEMBL29508878 0.80 KMT2A (0.71) KMT2AMEN1ALDH1A1HPGDLMNA
SCHEMBL297043 0.80 KMT2A (0.71) KMT2AMEN1ALDH1A1HPGDLMNA
SCHEMBL6642132 0.80 GAA (0.62) KMT2AMEN1CYP1A2CYP3A4ALDH1A1
SCHEMBL10604299 0.79 ALDH1A1 (0.66) KMT2AMEN1CYP1A2CYP3A4ALDH1A1
SCHEMBL8304862 0.79 GAA (0.76) KMT2AMEN1ALDH1A1HPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360802-A Antagonists of cholecystokinin and gastrin MERCK SHARPE & DOHME LTD. 1994-11-01 US disclosed
EP-0514133-A1 Benzodiazepine derivatives, compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1992-11-19 EP disclosed