SCHEMBL9301587

SCHEMBL9301587

Cc1ccccc1S(=O)(=O)NC(=O)c1cccc(NC(=O)N[C@]2(C3CCCCC3)N=Cc3ccccc3N(C)C2=O)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 10/20 0.57
CYSLTR1 Q9Y271 5/20 0.41
EPHX2 P34913 3/20 0.41
PPARG P37231 3/20 0.41
CYSLTR2 Q9NS75 3/20 0.38
MEN1 O00255 1/20 0.37
PTGES O14684 1/20 0.37
XPO1 O14980 1/20 0.37
SLC22A2 O15244 1/20 0.37
ABCC4 O15439 1/20 0.37
NR1I2 O75469 1/20 0.37
ABCB11 O95342 1/20 0.37
EGFR P00533 1/20 0.37
NR3C1 P04150 1/20 0.37
PGR P06401 1/20 0.37
POLB P06746 1/20 0.37
ADRA2A P08913 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
MAPT P10636 1/20 0.37
RARB P10826 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302356 0.92 CCKBR (0.48) CCKBRCYSLTR1EPHX2PPARGCYSLTR2
SCHEMBL9303126 0.90 CCKBR (0.55) CCKBRCYSLTR1EPHX2PPARGEGFR
SCHEMBL9301937 0.90 CCKBR (0.55) CCKBRCYSLTR1EPHX2PPARGEGFR
SCHEMBL9303570 0.90 CCKBR (0.45) CCKBRCYSLTR1EPHX2PPARGCYSLTR2
SCHEMBL9701161 0.87 CCKBR (0.55) CCKBRCCKARBACE1BACE2
SCHEMBL9702299 0.87 CCKBR (0.55) CCKBRCCKARBACE1BACE2
SCHEMBL9301948 0.81 CCKBR (0.41) CCKBRNPC1RAB9ACCKARBACE1
SCHEMBL9699964 0.80 CCKBR (0.45) CCKBRMAPTMAPK1TP53HTT
SCHEMBL9699961 0.80 CCKBR (0.45) CCKBRMAPTMAPK1TP53HTT
SCHEMBL9218194 0.75 CCKBR (0.35) CCKBRCCKARBACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0514133-A1 Benzodiazepine derivatives, compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1992-11-19 EP claimed
US-5360802-A Antagonists of cholecystokinin and gastrin MERCK SHARPE & DOHME LTD. 1994-11-01 US disclosed
EP-0514133-A1 Benzodiazepine derivatives, compositions containing them and their use in therapy MERCK SHARP & DOHME LTD. (GB) 1992-11-19 EP disclosed