SCHEMBL9301663

SCHEMBL9301663

CCCC(C(=O)OCC)c1cncc(C#Cc2cc3c(cc2C)OCCC3(C)C)n1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.34
HNF4A P41235 1/20 0.34
CYP3A4 P08684 1/20 0.32
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RARG P13631 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9304047 0.87 RARA (0.42) RXRAHNF4ACYP3A4RARARARB
SCHEMBL9302065 0.83 RARA (0.44) CYP3A4RARARARBRARGKMT2A
SCHEMBL9301695 0.83 RXRA (0.34) RXRAHNF4ACYP3A4RARARARB
SCHEMBL9302770 0.82 RXRA (0.37) RXRAHNF4ACYP3A4RARARARB
SCHEMBL9817739 0.80 RXRA (0.38) RXRAHNF4ACYP3A4RARARARB
SCHEMBL9139421 0.78 RXRA (0.37) RXRAHNF4ARARARARBRARG
SCHEMBL9301657 0.78 RXRA (0.34) RXRAHNF4ACYP3A4RARARARB
SCHEMBL9302638 0.77 CYP26A1 (0.38) RXRAHNF4ARARARARBRARG
SCHEMBL9304103 0.77 RARB (0.39) RXRAHNF4ACYP3A4RARARARB
SCHEMBL9302754 0.75 RXRA (0.36) RXRAHNF4ACYP3A4RARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed