SCHEMBL9302103

SCHEMBL9302103

CCOC(=O)CCCCc1cc(C#Cc2ccc3c(c2)C(C)(C)CCS3)cnn1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RARB P10826 11/20 0.56
RARG P13631 11/20 0.56
RARA P10276 10/20 0.56
CYP3A4 P08684 3/20 0.56
KMT2A Q03164 1/20 0.56
CYP26A1 O43174 2/20 0.47
RXRA P19793 2/20 0.35
CYP4F2 P78329 1/20 0.32
CYP4A11 Q02928 1/20 0.32
CRABP2 P29373 1/20 0.31
TBXAS1 P24557 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301902 0.89 CYP3A4 (0.53) RARBRARGRARACYP3A4KMT2A
SCHEMBL9303234 0.89 RARB (0.61) RARBRARGRARACYP3A4KMT2A
SCHEMBL9303655 0.88 CYP3A4 (0.43) RARBRARGRARACYP3A4KMT2A
SCHEMBL6664870 0.87 RARB (0.62) RARBRARGRARACYP3A4KMT2A
SCHEMBL6665899 0.86 RARB (0.62) RARBRARGRARACYP3A4KMT2A
SCHEMBL9673775 0.86 RARA (0.65) RARBRARGRARACYP3A4KMT2A
SCHEMBL9303289 0.85 RARA (0.59) RARBRARGRARACYP3A4KMT2A
SCHEMBL9817849 0.85 RARB (0.58) RARBRARGRARACYP3A4KMT2A
SCHEMBL9302100 0.83 RARA (0.53) RARBRARGRARACYP3A4KMT2A
SCHEMBL9302931 0.83 RARA (0.39) RARBRARGRARACYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed