SCHEMBL9817856

SCHEMBL9817856

CCOC(=O)CCCCc1ccc(C#Cc2ccc3c(c2)C(SC)(SC)CCO3)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4Z1 Q86W10 2/20 0.38
MGLL Q99685 2/20 0.37
FAAH O00519 1/20 0.37
ACACB O00763 3/20 0.35
CYP4F11 Q9HBI6 1/20 0.35
CYP4F12 Q9HCS2 1/20 0.35
CYP4F2 P78329 2/20 0.34
CYP4A11 Q02928 2/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
ALOX5 P09917 1/20 0.33
MAPT P10636 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
GLA P06280 1/20 0.33
RAB9A P51151 1/20 0.33
FFAR1 O14842 1/20 0.33
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9817683 0.97 CYP4Z1 (0.37) CYP4Z1MGLLFAAHACACBCYP4F11
SCHEMBL9817777 0.92 PPARA (0.35) CYP4Z1MGLLFAAHCYP4F2CYP4A11
SCHEMBL6671545 0.90 CYP3A4 (0.42) CYP4Z1MGLLFAAHACACBCYP4F2
SCHEMBL9817649 0.89 ALOX5 (0.36) CYP4Z1CYP4F11CYP4F12CYP4F2CYP4A11
SCHEMBL6668825 0.89 PRSS1 (0.33) CYP4Z1CYP4F2CYP4A11ALDH1A1NPC1
SCHEMBL9817759 0.88 CYP26A1 (0.40) CYP4Z1MGLLFAAHACACBCYP4F11
SCHEMBL6665905 0.88 CYP3A4 (0.37) CYP4F2CYP4A11ALDH1A1MAPTNPC1
SCHEMBL8668822 0.87 CYP4Z1 (0.39) CYP4Z1MGLLFAAHACACBCYP4F11
SCHEMBL6668884 0.87 CYP3A4 (0.32) CYP4F2CYP4A11ALDH1A1NPC1TP53
SCHEMBL9817635 0.87 CYP4F2 (0.41) MGLLFAAHCYP4F2CYP4A11FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290130-B1 ACETYLENES DISUBSTITUTED WITH A PHENYL GROUP AND A HETEROBICYCLIC GROUP HAVING RETINOID LIKE ACTIVITY ALLERGAN, INC (US) 1991-11-06 EP disclosed
US-4810804-A PSORIASIS ALLERGAN, INC. (US) 1989-03-07 US disclosed
EP-0290130-A1 Acetylenes disubstituted with a phenyl group and a heterobicyclic group having retinoid like activity ALLERGAN, INC (US) 1988-11-09 EP disclosed