SCHEMBL9302233

SCHEMBL9302233

O=c1cc2n(C3CC3)c3cc(N4CCNCC4)c(F)cc3n2c(=O)n1OCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
HSD17B10 Q99714 4/20 0.39
KDM4E B2RXH2 3/20 0.39
LMNA P02545 3/20 0.39
HPGD P15428 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
TOP2A P11388 1/20 0.39
TOP2B Q02880 1/20 0.39
HTR1A P08908 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 1/20 0.36
OPRL1 P41146 1/20 0.35
HTR6 P50406 3/20 0.34
TSHR P16473 2/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301963 0.90 ALDH1A1 (0.36) ALDH1A1KDM4ELMNAHPGDCYP1A2
SCHEMBL9302877 0.88 GRM5 (0.39) ALDH1A1HSD17B10KDM4ELMNAHPGD
SCHEMBL9301342 0.84 STS (0.38) LMNABRD4
SCHEMBL9302209 0.82 PIK3CD (0.35) ALDH1A1HSD17B10KDM4ELMNAHPGD
SCHEMBL9303648 0.79 ACE (0.34) CASP1CHRM4
SCHEMBL9301465 0.79 ALDH1A1 (0.45) ALDH1A1HSD17B10KDM4ELMNAHPGD
SCHEMBL9302936 0.79 ALDH1A1 (0.43) ALDH1A1HSD17B10KDM4ELMNAHPGD
Hydrochloric Acid SCHEMBL9304165 0.78 ALDH1A1 (0.45) ALDH1A1HSD17B10KDM4ELMNAHPGD
SCHEMBL9301603 0.76 ALDH1A1 (0.41) ALDH1A1HSD17B10KDM4ELMNAHPGD
SCHEMBL9301409 0.76 ALDH1A1 (0.41) ALDH1A1HSD17B10KDM4ELMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed