SCHEMBL9302877

SCHEMBL9302877

O=C(O)N1CCN(c2cc3c(cc2F)n2c(=O)n(OCc4ccccc4)c(=O)cc2n3C2CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.39
PIK3CG P48736 2/20 0.36
PIK3CD O00329 1/20 0.36
PIK3R1 P27986 1/20 0.36
PIK3CA P42336 1/20 0.36
ALDH1A1 P00352 6/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
HPGD P15428 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KDM4E B2RXH2 5/20 0.35
CHRM4 P08173 2/20 0.35
ALOX15 P16050 2/20 0.34
KMT2A Q03164 2/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GAA P10253 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301963 0.90 ALDH1A1 (0.36) GRM5PIK3CGPIK3CDPIK3R1PIK3CA
SCHEMBL9302233 0.88 ALDH1A1 (0.39) ALDH1A1HPGDKDM4ECHRM4KMT2A
SCHEMBL9302209 0.88 PIK3CD (0.35) GRM5PIK3CGPIK3CDPIK3R1PIK3CA
SCHEMBL9303648 0.81 ACE (0.34) CHRM4
SCHEMBL9847726 0.78 KDM4E (0.40) PIK3CGPIK3CDPIK3R1PIK3CAALDH1A1
SCHEMBL9303411 0.76 ALDH1A1 (0.41) GRM5ALDH1A1HPGDKDM4EKMT2A
SCHEMBL6799741 0.72 THRB (0.41) ALDH1A1HPGDKDM4ELMNAHSD17B10
SCHEMBL9302393 0.70 KDM4E (0.38) PIK3CGPIK3CDPIK3R1PIK3CAALDH1A1
SCHEMBL9302145 0.70 CRBN (0.38) ALDH1A1SMN1; SMN2HPGDKDM4EKMT2A
SCHEMBL9302286 0.69 OPRM1 (0.38) ALDH1A1SMN1; SMN2KDM4ELMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed