SCHEMBL9302209

SCHEMBL9302209

C[C@H](NC(=O)O)C(=O)N1CCN(c2cc3c(cc2F)n2c(=O)n(OCc4ccccc4)c(=O)cc2n3C2CC2)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.35
PIK3R1 P27986 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CG P48736 1/20 0.35
GRM5 P41594 1/20 0.34
ALDH1A1 P00352 7/20 0.34
KDM4E B2RXH2 7/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
HPGD P15428 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
LMNA P02545 4/20 0.33
HTT P42858 3/20 0.33
HSD17B10 Q99714 2/20 0.33
ALOX15 P16050 1/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302877 0.88 GRM5 (0.39) PIK3CDPIK3R1PIK3CAPIK3CGGRM5
SCHEMBL9301963 0.85 ALDH1A1 (0.36) PIK3CDPIK3R1PIK3CAPIK3CGGRM5
SCHEMBL9302233 0.82 ALDH1A1 (0.39) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL9303648 0.76 ACE (0.34)
SCHEMBL9302393 0.73 KDM4E (0.38) PIK3CDPIK3R1PIK3CAPIK3CGALDH1A1
SCHEMBL9303411 0.72 ALDH1A1 (0.41) GRM5ALDH1A1KDM4EHPGDMEN1
SCHEMBL9847726 0.69 KDM4E (0.40) PIK3CDPIK3R1PIK3CAPIK3CGALDH1A1
SCHEMBL9303155 0.68 HRH3 (0.38) ALDH1A1KDM4ESMN1; SMN2LMNAMAPT
SCHEMBL6799741 0.67 THRB (0.41) ALDH1A1KDM4EHPGDLMNAHSD17B10
SCHEMBL9302145 0.66 CRBN (0.38) ALDH1A1KDM4ESMN1; SMN2HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed