SCHEMBL9302591

SCHEMBL9302591

CC1(C)CCSc2ccc(C#Cc3cncc(CC(=O)O)n3)cc21

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RARB P10826 15/20 0.61
RARG P13631 15/20 0.61
RARA P10276 13/20 0.61
CYP3A4 P08684 3/20 0.61
CYP26A1 O43174 2/20 0.61
KMT2A Q03164 1/20 0.56
RXRA P19793 2/20 0.39
CRABP2 P29373 1/20 0.38
SSTR5 P35346 1/20 0.33
SLC22A12 Q96S37 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301486 0.88 RARB (0.56) RARBRARGRARACYP3A4CYP26A1
SCHEMBL9303919 0.88 RARA (0.64) RARBRARGRARACYP3A4CYP26A1
SCHEMBL6664613 0.85 CYP3A4 (0.67) RARBRARGRARACYP3A4CYP26A1
SCHEMBL6666821 0.85 CYP3A4 (0.64) RARBRARGRARACYP3A4CYP26A1
SCHEMBL9302702 0.83 RARA (0.41) RARBRARGRARACYP3A4CYP26A1
SCHEMBL9302949 0.82 CYP3A4 (0.57) RARBRARGRARACYP3A4CYP26A1
SCHEMBL6665585 0.81 CYP3A4 (0.64) RARBRARGRARACYP3A4CYP26A1
SCHEMBL6670285 0.81 CYP26A1 (0.73) RARBRARGRARACYP3A4CYP26A1
SCHEMBL9303289 0.81 RARA (0.59) RARBRARGRARACYP3A4CYP26A1
SCHEMBL9302953 0.80 CYP26A1 (0.45) RARBRARGRARACYP3A4CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed