SCHEMBL9302706

SCHEMBL9302706

ClCc1cccc(N2CCOCC2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGXT P21549 2/20 0.65
LMNA P02545 1/20 0.53
KMO O15229 1/20 0.51
SIGMAR1 Q99720 4/20 0.51
TMEM97 Q5BJF2 3/20 0.51
ADRA2A P08913 2/20 0.51
ADRA2B P18089 2/20 0.51
ADRA2C P18825 1/20 0.51
DRD4 P21917 2/20 0.48
HRH1 P35367 1/20 0.48
HTR2B P41595 1/20 0.48
AKR1C3 P42330 1/20 0.47
PLOD2 O00469 1/20 0.45
PLOD3 O60568 1/20 0.45
PLOD1 Q02809 1/20 0.45
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29867053 1.00 AGXT (0.65) AGXTLMNAKMOSIGMAR1TMEM97
SCHEMBL23662605 0.85 AGXT (0.63) AGXTLMNAKMOSIGMAR1TMEM97
SCHEMBL22964326 0.83 AGXT (0.65) AGXTLMNAKMOSIGMAR1TMEM97
SCHEMBL18295011 0.83 AGXT (0.65) AGXTLMNAKMOSIGMAR1TMEM97
SCHEMBL4507051 0.83 AGXT (0.65) AGXTLMNAKMOSIGMAR1TMEM97
SCHEMBL671148 0.83 AGXT (0.65) AGXTLMNAKMOSIGMAR1TMEM97
SCHEMBL108136 0.83 AGXT (0.69) AGXTLMNAKMOSIGMAR1TMEM97
SCHEMBL16726976 0.82 PRMT6 (0.63) AGXTSIGMAR1MEN1ALDH1A1MAPT
SCHEMBL27329825 0.81 LMNA (0.71) AGXTLMNAKMOAKR1C3PLOD2
SCHEMBL425652 0.80 AGXT (0.66) AGXTLMNAKMOSIGMAR1TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021143924-A1 BORIC ACID DERIVATIVE 首药控股(北京)股份有限公司 2021-07-22 WO disclosed
US-5281720-A Antiasthmatics, antiallergens, antiinflammatory agents and cytoprotective agents MERCK FROSST CANADA, INC. 1994-01-25 US disclosed
US-5227399-A Pyranylphenyl naphthalene lactones as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1993-07-13 US disclosed
EP-0501579-A1 Naphthalene lactones as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1992-09-02 EP disclosed
EP-0501578-A1 Pyranylphenyl hydroxyalkylnaphthoic acids as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA INC. (CA) 1992-09-02 EP disclosed