SCHEMBL9302794

SCHEMBL9302794

O=C1c2cc(Br)ccc2-c2nc(C=NO)ccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCL2 P10415 3/20 0.45
MCL1 Q07820 2/20 0.45
S100A4 P26447 2/20 0.43
PTPRC P08575 1/20 0.39
LCK P06239 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
MAPK1 P28482 1/20 0.34
EDNRB P24530 1/20 0.33
EDNRA P25101 1/20 0.33
TSHR P16473 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301644 0.82 S100A4 (0.48) BCL2MCL1S100A4PTPRCLCK
SCHEMBL9301758 0.72 S100A4 (0.52) BCL2MCL1S100A4PTPRCCA1
SCHEMBL9301771 0.72 BCL2 (0.49) BCL2MCL1S100A4PTPRCLCK
SCHEMBL9302326 0.69 S100A4 (0.47) BCL2MCL1S100A4PTPRCCA1
SCHEMBL762135 0.68 S100A4 (0.80) BCL2MCL1S100A4PTPRCLCK
SCHEMBL39700 0.68 S100A4 (0.90) BCL2MCL1S100A4PTPRCLCK
SCHEMBL29664078 0.68 S100A4 (0.80) BCL2MCL1S100A4PTPRCLCK
SCHEMBL3717374 0.68 S100A4 (0.80) BCL2MCL1S100A4PTPRCLCK
SCHEMBL29390614 0.68 S100A4 (0.90) BCL2MCL1S100A4PTPRCLCK
SCHEMBL9302996 0.66 GAA (0.60) BCL2MCL1S100A4PTPRCGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994009002-A1 2-(AZA-9-FLUORENONYL)CARBAPENEM ANTIBACTERIAL AGENTS MERCK & CO., INC. (US) 1994-04-28 WO disclosed
US-5294610-A Staphylococcus; side effect reduction MERCK & CO. INC. (US) 1994-03-15 US disclosed