SCHEMBL9303612

SCHEMBL9303612

N=C(N)c1ccc(NC(=O)c2ccccc2N=C(N)N)c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KDM4E B2RXH2 5/20 0.41
GAA P10253 2/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
PLAU P00749 2/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
SIGMAR1 Q99720 2/20 0.38
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303484 0.95 NPC1 (0.49) NPC1RAB9AKDM4EGAAMAPT
SCHEMBL9303327 0.82 RAB9A (0.44) NPC1RAB9AKDM4EGAAMAPT
SCHEMBL9303967 0.81 KCNJ11 (0.43) NPC1RAB9AKDM4EMAPTPLAU
SCHEMBL9303104 0.80 NPC1 (0.49) NPC1RAB9AKDM4EGAAMAPT
SCHEMBL9303554 0.80 NPC1 (0.46) NPC1RAB9AKDM4EGAAMAPT
SCHEMBL9303218 0.80 PLAU (0.44) NPC1RAB9AKDM4EMAPTPLAU
SCHEMBL9303439 0.78 NPC1 (0.45) NPC1RAB9AKDM4EGAAMAPT
SCHEMBL9303532 0.77 PLAU (0.57) NPC1RAB9APLAUCHRNB2CHRNB4
SCHEMBL9302787 0.77 PLAU (0.45) NPC1RAB9AMEN1KMT2APLAU
SCHEMBL9304147 0.77 DEGS1 (0.44) NPC1RAB9AMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5352704-A Antiviral agents BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-10-04 US disclosed
EP-0434432-B1 Guanidinobenzene derivatives BANYU PHARMA CO LTD (JP) 1994-05-04 EP disclosed
EP-0434432-A1 Guanidinobenzene derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1991-06-26 EP disclosed