SCHEMBL9303651

SCHEMBL9303651

CCOC(=O)CCCCc1nnccc1C#Cc1cc2c(cc1C)SCCC2(C)C

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RARA P10276 7/20 0.40
RARB P10826 7/20 0.40
RARG P13631 7/20 0.40
CYP3A4 P08684 2/20 0.40
KMT2A Q03164 1/20 0.40
TBXAS1 P24557 1/20 0.33
CYP26A1 O43174 1/20 0.32
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
RXRA P19793 1/20 0.31
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30
CYP4Z1 Q86W10 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302100 0.89 RARA (0.53) RARARARBRARGCYP3A4KMT2A
SCHEMBL9302045 0.86 RARA (0.41) RARARARBRARGCYP3A4KMT2A
SCHEMBL6668353 0.84 RARA (0.46) RARARARBRARGCYP3A4KMT2A
SCHEMBL9301685 0.83 RXRA (0.36) RARARARBRARGTBXAS1CYP4F2
SCHEMBL9303655 0.83 CYP3A4 (0.43) RARARARBRARGCYP3A4KMT2A
SCHEMBL6667776 0.82 RARA (0.47) RARARARBRARGCYP3A4KMT2A
SCHEMBL9302012 0.82 RARA (0.44) RARARARBRARGCYP3A4KMT2A
SCHEMBL6665864 0.81 RARA (0.39) RARARARBRARGCYP3A4KMT2A
SCHEMBL6668278 0.81 RARA (0.53) RARARARBRARGCYP3A4KMT2A
SCHEMBL9302053 0.81 CYP3A4 (0.43) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed