SCHEMBL9302100

SCHEMBL9302100

CCOC(=O)CCCCc1nnccc1C#Cc1ccc2c(c1)C(C)(C)CCS2

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RARA P10276 9/20 0.53
RARB P10826 9/20 0.53
RARG P13631 9/20 0.53
CYP3A4 P08684 3/20 0.53
KMT2A Q03164 1/20 0.53
CYP26A1 O43174 2/20 0.44
RXRA P19793 2/20 0.34
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
CRABP2 P29373 1/20 0.31
TBXAS1 P24557 1/20 0.30
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303651 0.89 RARA (0.40) RARARARBRARGCYP3A4KMT2A
SCHEMBL9303286 0.85 RARB (0.56) RARARARBRARGCYP3A4KMT2A
SCHEMBL9302925 0.84 RARA (0.36) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817849 0.83 RARB (0.58) RARARARBRARGCYP3A4KMT2A
SCHEMBL9302103 0.83 RARB (0.56) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817631 0.83 RARA (0.54) RARARARBRARGCYP3A4KMT2A
SCHEMBL6665899 0.83 RARB (0.62) RARARARBRARGCYP3A4KMT2A
SCHEMBL6664870 0.82 RARB (0.62) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817773 0.81 RARA (0.55) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817673 0.81 RARB (0.58) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed