SCHEMBL9304071

SCHEMBL9304071

CCOC(=O)Cc1cncc(C#Cc2ccc3c(c2)C(C)(C)CCO3)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 8/20 0.44
RARB P10826 8/20 0.44
RARG P13631 8/20 0.44
CYP3A4 P08684 3/20 0.44
KMT2A Q03164 1/20 0.44
CYP26A1 O43174 3/20 0.36
RXRA P19793 2/20 0.36
CYP26B1 Q9NR63 1/20 0.36
HNF4A P41235 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
MAPT P10636 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
CRABP2 P29373 1/20 0.33
TP53 P04637 1/20 0.32
GLA P06280 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9304041 0.89 RARA (0.41) RARARARBRARGCYP3A4KMT2A
SCHEMBL9303922 0.89 CYP3A4 (0.37) RARARARBRARGCYP3A4KMT2A
SCHEMBL9302953 0.88 CYP26A1 (0.45) RARARARBRARGCYP3A4KMT2A
SCHEMBL9303176 0.84 RARB (0.41) RARARARBRARGCYP3A4KMT2A
SCHEMBL9302760 0.83 RARA (0.46) RARARARBRARGCYP3A4KMT2A
SCHEMBL9303919 0.82 RARA (0.64) RARARARBRARGCYP3A4KMT2A
SCHEMBL9817608 0.81 RARA (0.42) RARARARBRARGCYP3A4KMT2A
SCHEMBL9304047 0.81 RARA (0.42) RARARARBRARGCYP3A4KMT2A
SCHEMBL9304108 0.80 RARA (0.39) RARARARBRARGCYP3A4KMT2A
SCHEMBL9137701 0.80 RARB (0.41) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed