SCHEMBL9304041

SCHEMBL9304041

CCOC(=O)CCCCc1cncc(C#Cc2ccc3c(c2)C(C)(C)CCO3)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 7/20 0.41
RARB P10826 7/20 0.41
RARG P13631 7/20 0.41
CYP3A4 P08684 3/20 0.41
KMT2A Q03164 1/20 0.41
RXRA P19793 2/20 0.34
HNF4A P41235 1/20 0.34
CYP26A1 O43174 3/20 0.32
CYP26B1 Q9NR63 1/20 0.32
TBXAS1 P24557 1/20 0.32
NPSR1 Q6W5P4 2/20 0.32
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
PTGER4 P35408 1/20 0.31
CYP4F2 P78329 1/20 0.31
CYP4A11 Q02928 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303290 0.90 CYP3A4 (0.35) RARARARBRARGCYP3A4KMT2A
SCHEMBL9304071 0.89 RARA (0.44) RARARARBRARGCYP3A4KMT2A
SCHEMBL9304108 0.89 RARA (0.39) RARARARBRARGCYP3A4KMT2A
SCHEMBL6684655 0.88 RARA (0.46) RARARARBRARGCYP3A4KMT2A
SCHEMBL9301657 0.87 RXRA (0.34) RARARARBRARGCYP3A4KMT2A
SCHEMBL6667261 0.87 RARA (0.44) RARARARBRARGCYP3A4KMT2A
SCHEMBL9302931 0.85 RARA (0.39) RARARARBRARGCYP3A4KMT2A
SCHEMBL6669569 0.85 RARA (0.43) RARARARBRARGCYP3A4KMT2A
SCHEMBL6669581 0.84 RARA (0.49) RARARARBRARGCYP3A4KMT2A
SCHEMBL9303289 0.84 RARA (0.59) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed