SCHEMBL9304331

SCHEMBL9304331

CCOC(=O)Cc1cc(C#Cc2cc3c(cc2C)OCCC3(C)C)cnn1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.36
HNF4A P41235 1/20 0.36
RARA P10276 3/20 0.33
RARB P10826 3/20 0.33
RARG P13631 3/20 0.33
CYP3A4 P08684 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
CYP26A1 O43174 1/20 0.31
CYP26B1 Q9NR63 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301689 0.89 RXRA (0.35) RXRAHNF4ARARARARBRARG
SCHEMBL9302749 0.89 CYP26A1 (0.38) RXRAHNF4ARARARARBRARG
SCHEMBL9303176 0.87 RARB (0.41) RXRAHNF4ARARARARBRARG
SCHEMBL9301379 0.85 RXRA (0.40) RXRAHNF4ARARARARBRARG
SCHEMBL9817887 0.82 RXRA (0.41) RXRAHNF4ARARARARBRARG
SCHEMBL9302684 0.82 RARA (0.46) RXRARARARARBRARGCYP3A4
SCHEMBL9303121 0.81 RXRA (0.34) RXRAHNF4ARARARARBRARG
SCHEMBL9301695 0.81 RXRA (0.34) RXRAHNF4ARARARARBRARG
SCHEMBL9302689 0.80 NPC1 (0.32) NPC1MAPTRAB9ASMN1; SMN2NPSR1
SCHEMBL6671507 0.78 RXRA (0.37) RXRAHNF4ARARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354752-A A dimethylthiochroman or dimethylchroman-6-yl-ethynyl-pyridazin- or pyrimidin- or pyrazin-for treating skin disorders psoriasis ALLERGAN, INC. (US) 1994-10-11 US claimed