SCHEMBL9304621

SCHEMBL9304621

NCCCCn1nc(-c2ccc(Cl)c(Cl)c2)c2cnccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TEAD2 Q15562 1/20 0.43
MERTK Q12866 3/20 0.38
HASPIN Q8TF76 1/20 0.36
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 2/20 0.34
CYP3A4 P08684 2/20 0.34
HRH1 P35367 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
RPS6KA5 O75582 1/20 0.34
P2RX7 Q99572 1/20 0.34
ESR1 P03372 1/20 0.34
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34
MAOA P21397 4/20 0.33
MAOB P27338 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303543 0.96 TEAD2 (0.39) TEAD2MERTKHASPINKDM4EHSD17B10
SCHEMBL9303594 0.92 HRH1 (0.36) TEAD2KDM4EHSD17B10CYP3A4HRH1
SCHEMBL9305127 0.88 MERTK (0.41) MERTKHASPINKDM4EHSD17B10CYP3A4
Fumaric Acid SCHEMBL8138733 0.88 TEAD2 (0.40) TEAD2KDM4EHSD17B10TSHRESR1
Maleic Acid SCHEMBL8138730 0.88 TEAD2 (0.40) TEAD2KDM4EHSD17B10TSHRESR1
SCHEMBL9257304 0.85 MERTK (0.44) MERTKHASPINKDM4EHSD17B10HRH1
SCHEMBL8135725 0.84 LTA4H (0.39) MERTKKDM4EHSD17B10CYP3A4ALDH1A1
Maleic Acid SCHEMBL8135697 0.83 TEAD2 (0.37) TEAD2KDM4EHSD17B10TSHRNAMPT
Fumaric Acid SCHEMBL8135703 0.83 TEAD2 (0.37) TEAD2KDM4EHSD17B10TSHRNAMPT
SCHEMBL9304792 0.81 MAPK13 (0.41) MERTKKDM4EHSD17B10TSHRRPS6KA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US claimed