SCHEMBL9304715

SCHEMBL9304715

[CH]1CCNC[C]1c1cccc2ccccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.42
CYP2D6 P10635 2/20 0.38
HTR2A P28223 2/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
CYP1A2 P05177 1/20 0.38
HTR1A P08908 1/20 0.38
NCF1 P14598 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR7 P34969 1/20 0.38
MTOR P42345 1/20 0.38
HTR3A P46098 1/20 0.38
HTR5A P47898 1/20 0.38
HTR6 P50406 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25171978 0.76 HTR2A (0.50) NISCHCYP2D6HTR2AHTR3EHTR3B
SCHEMBL8292046 0.74 GSK3A (0.40) CYP2D6HTR2ACYP1A2PRCPHTR2C
SCHEMBL4718750 0.68 RYR2 (0.42) NISCHCYP2D6HTR2AHTR3EHTR3B
SCHEMBL894789 0.68 NISCH (0.57) NISCHCYP2D6HTR2AHTR3EHTR3B
SCHEMBL27953 0.67 ALDH1A1 (0.59) NISCHCYP1A2TSHRNFKB1HSD17B10
SCHEMBL25302086 0.67 ALDH1A1 (0.59) NISCHCYP1A2TSHRNFKB1HSD17B10
SCHEMBL29350007 0.67 ALDH1A1 (0.59) NISCHCYP1A2TSHRNFKB1HSD17B10
SCHEMBL9044714 0.67 NISCH (0.47) NISCHCYP2D6HTR2AHTR3EHTR3B
SCHEMBL4765544 0.66 NISCH (0.55) NISCHCYP2D6HTR2AHTR3EHTR3B
SCHEMBL5408922 0.66 NISCH (0.39) NISCHCYP1A2HTR1ATSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0398413-A1 \"3,4-dehydropiperidine derivatives having psychotropic activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1990-11-22 EP claimed
US-5296497-A 3,4-dehydropiperidine derivatives having psychotropic activity DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1994-03-22 US disclosed
EP-0398413-A1 \"3,4-dehydropiperidine derivatives having psychotropic activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1990-11-22 EP disclosed