SCHEMBL9306032

SCHEMBL9306032

CC(C)(C)CC(C)(C)c1ccc2nc(S)oc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SHBG P04278 1/20 0.39
MAPT P10636 3/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP3A4 P08684 3/20 0.35
CYP2D6 P10635 1/20 0.35
HIF1A Q16665 1/20 0.35
CSNK1D P48730 1/20 0.33
CSNK1G2 P78368 1/20 0.33
SMN1; SMN2 Q16637 4/20 0.33
USP2 O75604 2/20 0.32
HDAC6 Q9UBN7 1/20 0.32
MEN1 O00255 1/20 0.32
ESR1 P03372 1/20 0.32
TP53 P04637 1/20 0.32
PGR P06401 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
AR P10275 1/20 0.32
DRD1 P21728 1/20 0.32
PTGS1 P23219 1/20 0.32
SLC6A2 P23975 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9308324 0.82 SHBG (0.39) SHBGMAPTKDM4ECYP3A4CYP2D6
SCHEMBL31208302 0.76 BACE1 (0.42) KDM4ESMN1; SMN2KCNH2
SCHEMBL18755165 0.76 BACE1 (0.42) KDM4ESMN1; SMN2KCNH2
SCHEMBL9305789 0.73 MAPT (0.35) SHBGMAPTHDAC6TP53
SCHEMBL9305794 0.71 HDAC4 (0.33) SHBGMAPTCYP3A4CYP2D6HIF1A
SCHEMBL18174921 0.70 SMN1; SMN2 (0.43) MAPTKDM4ECYP3A4CYP2D6SMN1; SMN2
SCHEMBL23743981 0.70 SMN1; SMN2 (0.41) MAPTKDM4ECSNK1DCSNK1G2SMN1; SMN2
SCHEMBL9304978 0.70 SCN10A (0.43) SHBGMAPTCYP3A4CYP2D6CSNK1D
SCHEMBL9304946 0.70 CSNK1D (0.40) SHBGMAPTCYP3A4CYP2D6HIF1A
SCHEMBL2538594 0.70 KDM4E (0.59) MAPTKDM4ECYP3A4CYP2D6SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed