SCHEMBL9304978

SCHEMBL9304978

CC(C)(C)CC(C)(C)c1ccc2nc(S)[nH]c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 11/20 0.43
KCNH2 Q12809 1/20 0.43
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HSD17B10 Q99714 1/20 0.40
SHBG P04278 1/20 0.39
METAP2 P50579 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2E1 P05181 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C8 P10632 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2B6 P20813 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPBWR1 P48145 1/20 0.37
PDE10A Q9Y233 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
PLK4 O00444 1/20 0.36
CHEK1 O14757 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9304989 0.88 SHBG (0.39) SCN10AKCNH2MAPTSHBGCYP1A2
SCHEMBL29213213 0.82 SCN10A (0.61) SCN10AKCNH2METAP2PDE10ATRPV1
SCHEMBL9303891 0.82 SCN10A (0.43) SCN10AKCNH2GAAMAPTHSD17B10
SCHEMBL10579210 0.78 SCN10A (0.38) SCN10AKCNH2GAAMAPTHSD17B10
SCHEMBL2107034 0.76 NPBWR1 (0.58) SCN10AKCNH2GAAMAPTHSD17B10
SCHEMBL20348683 0.72 KIF11 (0.53) KCNH2MAPTSHBGCYP3A4CYP2D6
SCHEMBL9303902 0.70 SHBG (0.39) SCN10AKCNH2GAAMAPTSHBG
SCHEMBL9304946 0.70 CSNK1D (0.40) KCNH2GAAMAPTSHBGCYP3A4
SCHEMBL9306032 0.70 SHBG (0.39) KCNH2MAPTSHBGCYP3A4CYP2D6
SCHEMBL229608 0.70 KMT2A (0.58) GAAMAPTHSD17B10METAP2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0161220-B1 PROCESS FOR THE PREPARATION OF BETA-(BENZOTHIAZOLYLTHIO) AND BETA (BENZIMIDAZOLYLTHIO)CARBOXYLIC-ACID DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-14 EP disclosed
US-4652653-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio)-carboxylic acid derivatives CIBA-GEIGY CORPORATION (US) 1987-03-24 US disclosed
US-4612378-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio-carboxylic acids CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed
EP-0161220-A2 Process for the preparation of beta-(benzothiazolylthio) and beta (benzimidazolylthio)carboxylic-acid derivatives CIBA-GEIGY AG (CH) 1985-11-13 EP disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed
EP-0126030-A2 Process for the preparation of beta-(benzothiazolylthio) and beta-(benzimidazolylthio) carboxylic acids CIBA-GEIGY AG (CH) 1984-11-21 EP disclosed