SCHEMBL9306089

SCHEMBL9306089

CCCCCCCCCCCCCCOc1cccc(CN(Cc2ccccn2)S(=O)(=O)c2ccc(C)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.52
CA1 P00915 3/20 0.52
CA2 P00918 3/20 0.52
CA4 P22748 3/20 0.52
CA9 Q16790 3/20 0.52
PDE4A P27815 1/20 0.52
PDE4B Q07343 1/20 0.52
PDE4C Q08493 1/20 0.52
PDE4D Q08499 1/20 0.52
CNR2 P34972 3/20 0.50
KCNA5 P22460 1/20 0.50
KMT2A Q03164 1/20 0.49
CXCR3 P49682 7/20 0.48
MAPK1 P28482 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TAS2R14 Q9NYV8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL9306886 0.81 CA12 (0.48) CA12CA1CA2CA4CA9
SCHEMBL12863045 0.80 KMT2A (0.72) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL16908049 0.79 KMT2A (0.77) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL9308313 0.76 CYP2D6 (0.47) CNR2
SCHEMBL9308959 0.74 CXCR3 (0.48) PDE4APDE4BPDE4CPDE4DKCNA5
SCHEMBL20393918 0.73 KMT2A (0.72) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL12863387 0.72 CXCR3 (0.69) PDE4APDE4BPDE4CPDE4DCNR2
SCHEMBL12863586 0.70 CXCR3 (0.78) PDE4APDE4BPDE4CPDE4DCNR2
Iodide SCHEMBL9307636 0.70 CNR2 (0.46) CA12CA1CA2CA4CA9
SCHEMBL13649423 0.70 CXCR3 (0.71) CA12CA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5328921-A Antagonist of platelet activating factor AMERICAN CYANAMID COMPANY (US) 1994-07-12 US disclosed
US-5208247-A Antianaphylactic agents or septic shock AMERICAN CYANAMID COMPANY (US) 1993-05-04 US disclosed
EP-0530444-A1 Aryl, amide, imide, and carbamate pyridine antagonists of platelet activating factor AMERICAN CYANAMID COMPANY (US) 1993-03-10 EP disclosed