SCHEMBL9306708

SCHEMBL9306708

NC(=O)c1ccc2sc(S)nc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
DYRK1A Q13627 5/20 0.44
HDAC6 Q9UBN7 3/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
ATM Q13315 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
LCK P06239 1/20 0.40
KMT2A Q03164 1/20 0.39
GFER P55789 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
ILK Q13418 1/20 0.39
GLA P06280 1/20 0.38
KDM4B O94953 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6275004 0.87 DYRK1A (0.58) NPC1RAB9ASMN1; SMN2DYRK1AKDM4E
SCHEMBL2031602 0.85 NPC1 (0.68) NPC1RAB9ASMN1; SMN2HDAC6KDM4E
SCHEMBL19029338 0.81 NPC1 (0.50) NPC1RAB9ASMN1; SMN2DYRK1AHDAC6
SCHEMBL24052275 0.80 NPC1 (0.76) NPC1RAB9ASMN1; SMN2DYRK1AALDH1A1
SCHEMBL1748371 0.80 NPC1 (0.49) NPC1RAB9ASMN1; SMN2DYRK1AHDAC6
SCHEMBL9734141 0.80 THRB (0.56) NPC1RAB9ASMN1; SMN2DYRK1AHDAC6
SCHEMBL9305296 0.80 PIK3CA (0.50) NPC1RAB9ASMN1; SMN2HDAC6KDM4E
SCHEMBL10760937 0.77 NPC1 (0.47) NPC1RAB9ASMN1; SMN2DYRK1AHDAC6
SCHEMBL30874473 0.76 NPC1 (0.45) NPC1RAB9ASMN1; SMN2DYRK1AHDAC6
SCHEMBL10880169 0.76 NPC1 (0.52) NPC1RAB9ASMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
EP-0161220-B1 PROCESS FOR THE PREPARATION OF BETA-(BENZOTHIAZOLYLTHIO) AND BETA (BENZIMIDAZOLYLTHIO)CARBOXYLIC-ACID DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-14 EP disclosed
EP-0129506-B1 HETEROCYCLICALLY SUBSTITUTED THIO(CYCLO)ALKANE POLYCARBOXYLIC ACIDS CIBA-GEIGY AG (CH) 1991-03-06 EP disclosed
US-4652653-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio)-carboxylic acid derivatives CIBA-GEIGY CORPORATION (US) 1987-03-24 US disclosed
US-4612378-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio-carboxylic acids CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed
EP-0161220-A2 Process for the preparation of beta-(benzothiazolylthio) and beta (benzimidazolylthio)carboxylic-acid derivatives CIBA-GEIGY AG (CH) 1985-11-13 EP disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed
EP-0126030-A2 Process for the preparation of beta-(benzothiazolylthio) and beta-(benzimidazolylthio) carboxylic acids CIBA-GEIGY AG (CH) 1984-11-21 EP disclosed