SCHEMBL9306764

SCHEMBL9306764

CCCOc1cc(C)c(C)c2nc(S)sc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.37
KDM4E B2RXH2 2/20 0.37
HSD17B10 Q99714 1/20 0.37
MCHR1 Q99705 1/20 0.35
LMNA P02545 3/20 0.34
HTT P42858 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
MAPT P10636 3/20 0.34
TSHR P16473 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
ALDH1A1 P00352 2/20 0.33
HPGD P15428 1/20 0.33
PDE5A O76074 1/20 0.33
TLR8 Q9NR97 1/20 0.32
PPARG P37231 1/20 0.32
GAA P10253 2/20 0.32
MCOLN3 Q8TDD5 1/20 0.32
POLB P06746 1/20 0.32
ALOX5 P09917 2/20 0.31
NOS3 P29474 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9799959 0.83 MAPK1 (0.34) MAPK1KDM4EHSD17B10MCHR1LMNA
SCHEMBL9305425 0.71 MAPT (0.37) MAPK1KDM4EMCHR1LMNAHTT
SCHEMBL9304640 0.71 ALDH1A1 (0.35) MAPK1KDM4EMCHR1LMNAHTT
SCHEMBL13475555 0.70 HTT (0.51) MAPK1KDM4EHSD17B10MCHR1LMNA
SCHEMBL2095483 0.69 KDM4E (0.46) MAPK1KDM4EHSD17B10MAPTTSHR
SCHEMBL6691012 0.69 ALDH1A1 (0.54) MAPK1KDM4EMCHR1HTTMAPT
SCHEMBL9304646 0.69 ALDH1A1 (0.35) MAPK1KDM4EMCHR1LMNAHTT
SCHEMBL19122394 0.66 HTT (0.49) MAPK1KDM4EHSD17B10MCHR1LMNA
SCHEMBL9306412 0.66 MAPT (0.37) MAPK1KDM4EMCHR1LMNAHTT
SCHEMBL9306648 0.66 SMN1; SMN2 (0.34) MAPK1KDM4EMCHR1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
EP-0161220-B1 PROCESS FOR THE PREPARATION OF BETA-(BENZOTHIAZOLYLTHIO) AND BETA (BENZIMIDAZOLYLTHIO)CARBOXYLIC-ACID DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-14 EP disclosed
EP-0129506-B1 HETEROCYCLICALLY SUBSTITUTED THIO(CYCLO)ALKANE POLYCARBOXYLIC ACIDS CIBA-GEIGY AG (CH) 1991-03-06 EP disclosed
US-4652653-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio)-carboxylic acid derivatives CIBA-GEIGY CORPORATION (US) 1987-03-24 US disclosed
US-4612378-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio-carboxylic acids CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed
EP-0161220-A2 Process for the preparation of beta-(benzothiazolylthio) and beta (benzimidazolylthio)carboxylic-acid derivatives CIBA-GEIGY AG (CH) 1985-11-13 EP disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed
EP-0126030-A2 Process for the preparation of beta-(benzothiazolylthio) and beta-(benzimidazolylthio) carboxylic acids CIBA-GEIGY AG (CH) 1984-11-21 EP disclosed