SCHEMBL9305425

SCHEMBL9305425

CCCOc1cc(C)c(C)c2nc(S)oc12

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.37
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 3/20 0.37
HPGD P15428 2/20 0.37
LMNA P02545 4/20 0.36
HTT P42858 3/20 0.36
MCHR1 Q99705 1/20 0.35
MCOLN3 Q8TDD5 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
NPSR1 Q6W5P4 3/20 0.34
TSHR P16473 2/20 0.34
MAPK1 P28482 2/20 0.33
CA9 Q16790 3/20 0.32
TLR8 Q9NR97 1/20 0.32
GAA P10253 2/20 0.32
POLB P06746 1/20 0.32
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9306412 0.83 MAPT (0.37) MAPTALDH1A1KDM4EHPGDLMNA
SCHEMBL11094361 0.74 NUDT1 (0.32)
SCHEMBL9304640 0.71 ALDH1A1 (0.35) MAPTALDH1A1KDM4EHPGDLMNA
SCHEMBL9306764 0.71 MAPK1 (0.37) MAPTALDH1A1KDM4EHPGDLMNA
SCHEMBL13475555 0.70 HTT (0.51) MAPTALDH1A1KDM4EHPGDLMNA
SCHEMBL9304646 0.69 ALDH1A1 (0.35) MAPTALDH1A1KDM4EHPGDLMNA
SCHEMBL19122394 0.66 HTT (0.49) MAPTALDH1A1KDM4EHPGDLMNA
SCHEMBL9306648 0.66 SMN1; SMN2 (0.34) MAPTALDH1A1KDM4EHPGDLMNA
SCHEMBL9799959 0.66 MAPK1 (0.34) MAPTALDH1A1KDM4EHPGDLMNA
SCHEMBL29712144 0.64 HTT (0.46) MAPTALDH1A1KDM4EHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed