SCHEMBL9307018

SCHEMBL9307018

CS(=O)(=O)Nc1cccc([O])c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.59
ALDH1A1 P00352 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
POLB P06746 1/20 0.54
KIF11 P52732 1/20 0.50
NPC1 O15118 1/20 0.49
JAK2 O60674 1/20 0.49
RAB9A P51151 1/20 0.49
KDM1A O60341 1/20 0.49
NR3C1 P04150 1/20 0.49
BRD4 O60885 4/20 0.47
HSD17B1 P14061 1/20 0.47
HSD17B2 P37059 1/20 0.47
USP2 O75604 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL698855 0.87 KEAP1 (0.70) KEAP1ALDH1A1SMN1; SMN2POLBKIF11
SCHEMBL1488105 0.79 KEAP1 (0.59) KEAP1ALDH1A1SMN1; SMN2POLBKIF11
SCHEMBL9865360 0.79 KEAP1 (0.59) KEAP1ALDH1A1SMN1; SMN2POLBKIF11
SCHEMBL169803 0.79 KEAP1 (0.59) KEAP1ALDH1A1SMN1; SMN2POLBKIF11
SCHEMBL391197 0.78 KEAP1 (0.57) KEAP1ALDH1A1SMN1; SMN2POLBKIF11
SCHEMBL9770251 0.78 KEAP1 (0.57) KEAP1ALDH1A1SMN1; SMN2POLBKIF11
SCHEMBL1488101 0.78 KEAP1 (0.57) KEAP1ALDH1A1SMN1; SMN2POLBKIF11
SCHEMBL12811024 0.78 PTGS1 (0.57) KEAP1ALDH1A1SMN1; SMN2POLBKIF11
SCHEMBL9307026 0.78 HSD17B2 (0.67) KEAP1ALDH1A1SMN1; SMN2POLBKIF11
SCHEMBL10293008 0.78 KEAP1 (0.57) KEAP1ALDH1A1SMN1; SMN2POLBKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5284958-A Acylation, cyclization of a 5-hydrazine-1H-pyrazole FUJI PHOTO FILM CO., LTD. (JP) 1994-02-08 US disclosed
US-5214149-A Process for producing a 1H-pyrazolo[5,1-c]-1,2,4-triazole compound FUJI PHOTO FILM CO., LTD. (JP) 1993-05-25 US disclosed
EP-0127162-B1 COLOR PHOTOGRAPHIC LIGHT-SENSITIVE MATERIAL FUJI PHOTO FILM CO., LTD. (JP) 1989-11-15 EP disclosed
US-4842985-A COUPLER HAVING DYE MOIETY WITH SHIFTED MAXIMUM ABSORPTION WAVELENGTH, HUE-FIXING COMPOUND FUJI PHOTO FILM CO., LTD. (JP) 1989-06-27 US disclosed
US-4585728-A 2-EQUIVALENT MAGENTA COUPLER AND AMINE FUJI PHOTO FILM CO., LTD. (JP) 1986-04-29 US disclosed
US-4555479-A CONTAINING 5-PYRAZOLONE TYPE MAGENTA COUPLERS AND NITROGEN COMPOUND-PREVENTION STAINING FUJI PHOTO FILM CO., LTD. (JP) 1985-11-26 US disclosed
EP-0127162-A2 Color photographic light-sensitive material FUJI PHOTO FILM CO., LTD. (JP) 1984-12-05 EP disclosed
US-4477558-A CYAN DYES-FORMING COUPLERS; COLORFASTNESS FUJI PHOTO FILM CO., LTD. (JP) 1984-10-16 US disclosed