SCHEMBL9307067

SCHEMBL9307067

CCOC(=O)N1CCC(Cc2nc3ccccc3n2Cc2cccc(C)n2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.44
TSHR P16473 2/20 0.44
KDM4E B2RXH2 2/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
ATM Q13315 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
BRD4 O60885 3/20 0.42
ALDH1A2 O94788 2/20 0.42
ALDH2 P05091 2/20 0.42
ALDH3A1 P30838 2/20 0.42
ALDH1A3 P47895 2/20 0.42
GRIN2B Q13224 1/20 0.41
P2RX3 P56373 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CYP1A2 P05177 1/20 0.41
GRM5 P41594 1/20 0.41
NOS2 P35228 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538121 0.84 KDM4E (0.42) ALDH1A1TSHRKDM4EMAPTHPGD
Hydrochloric Acid SCHEMBL9537163 0.84 KDM4E (0.42) ALDH1A1TSHRKDM4EMAPTHPGD
SCHEMBL9537827 0.82 TSHR (0.46) ALDH1A1TSHRKDM4EMAPTHPGD
Hydrochloric Acid SCHEMBL9537839 0.81 HSD17B10 (0.52) ALDH1A1TSHRKDM4EMAPTHPGD
SCHEMBL9536891 0.81 ALDH1A1 (0.47) ALDH1A1TSHRKDM4EMAPTHPGD
SCHEMBL8561156 0.81 ALDH1A1 (0.42) ALDH1A1TSHRKDM4EMAPTHPGD
SCHEMBL9537236 0.81 MAPT (0.50) ALDH1A1TSHRKDM4EMAPTHPGD
SCHEMBL8138405 0.81 MEN1 (0.51) ALDH1A1MAPTSMN1; SMN2CYP1A2MEN1
SCHEMBL14173582 0.80 KCNH2 (0.50) NOS2MEN1KMT2A
SCHEMBL9382951 0.79 BRD4 (0.41) ALDH1A1TSHRKDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360807-A Substituted thiazolyl and substituted pyridinyl derivatives JANSSEN PHARMACEUTICA N.V. (BF) 1994-11-01 US disclosed
EP-0539420-A1 NOVEL SUBSTITUTED THIAZOLYL AND SUBSTITUTED PYRIDINYL DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1993-05-05 EP disclosed
WO-1992001697-A1 NOVEL SUBSTITUTED THIAZOLYL AND SUBSTITUTED PYRIDINYL DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1992-02-06 WO disclosed