SCHEMBL9307576

SCHEMBL9307576

CC1=C(C)C(=O)C(C(CCCCCC(=O)NCC(=O)OCc2ccccc2)c2ccccc2)=C(C)C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
ABCC3 O15438 1/20 0.41
NR1I2 O75469 1/20 0.41
ABCB11 O95342 1/20 0.41
NR3C1 P04150 1/20 0.41
RARG P13631 1/20 0.41
CNR1 P21554 1/20 0.41
OPRK1 P41145 1/20 0.41
NR1H2 P55055 1/20 0.41
PPARA Q07869 1/20 0.41
NR1H3 Q13133 1/20 0.41
NR1I3 Q14994 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9309809 0.85 FAAH (0.45) MEN1KMT2AHDAC3HDAC1HDAC2
SCHEMBL7833657 0.80 HDAC1 (0.49) CYP3A4NR1I2HDAC3HDAC1HDAC2
SCHEMBL9310852 0.80 PTPRC (0.43) PPARAHDAC3HDAC1HDAC2HDAC8
SCHEMBL9019233 0.80 PTPRC (0.43) PPARAHDAC3HDAC1HDAC2HDAC8
SCHEMBL9309807 0.79 HDAC1 (0.49) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL7831153 0.78 HDAC1 (0.44) ALDH1A1HPGDHDAC3HDAC1HDAC2
SCHEMBL7829363 0.78 HDAC3 (0.44) ALDH1A1CYP3A4CYP2D6CYP2C19HDAC3
SCHEMBL7831731 0.77 HDAC2 (0.46) ALDH1A1HDAC3HDAC1HDAC2HDAC8
SCHEMBL9308117 0.77 TBXAS1 (0.52) ALDH1A1HDAC3HDAC1HDAC2HDAC8
Seratrodast SCHEMBL98403 0.77 TBXAS1 (0.52) ALDH1A1HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304658-A Quinone derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-04-19 US disclosed
US-5180742-A Lipoxygenase Inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-19 US disclosed
EP-0232089-B1 QUINONE AMIDES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1991-03-13 EP disclosed
EP-0232089-A2 Quinone amides, their production and use Takeda Chemical Industries, Ltd. (JP) 1987-08-12 EP disclosed