SCHEMBL9309316

SCHEMBL9309316

O=Cc1ccn(-c2ccc(Cl)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.50
NOTUM Q6P988 3/20 0.40
MGLL Q99685 1/20 0.39
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38
TUBA1A Q71U36 1/20 0.38
TUBA1C Q9BQE3 1/20 0.38
TUBB6 Q9BUF5 1/20 0.38
TUBB2B Q9BVA1 1/20 0.38
TUBB1 Q9H4B7 1/20 0.38
GRIA1 P42261 1/20 0.36
GRIA2 P42262 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3095401 0.81 FAAH (0.39) MGLLGRIA1GRIA2GRIA3GRIA4
SCHEMBL6052596 0.81 MGLL (0.39) NOTUMMGLLTUBB4ATUBBTUBA3C
SCHEMBL7016863 0.81 CYP2A6 (0.50) NOTUMMGLLTUBB4ATUBBTUBA3C
SCHEMBL5126021 0.81 FAAH (0.39) HSD17B10MGLLGRIA1GRIA2GRIA3
SCHEMBL5126073 0.80 IDO1 (0.47) HSD17B10NOTUMMGLLTUBB4ATUBB
SCHEMBL1680730 0.80 COMT (0.48) MGLLTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL6630210 0.78 MEN1 (0.43) MGLLGRIA1GRIA2GRIA3GRIA4
SCHEMBL14395511 0.77 BCHE (0.39) GRIA1GRIA2GRIA3GRIA4ALDH1A1
SCHEMBL4118733 0.77 GRIA1 (0.46) GRIA1GRIA2GRIA3GRIA4HDAC2
SCHEMBL5129468 0.77 HDAC2 (0.37) NOTUMGRIA1GRIA2GRIA3GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242426-B1 GAMMA-HYDROXY-2-(FLUOROALKYLAMINOCARBONYL)-1-PIPERAZINEPENTANAMIDES AS HIV PROTEASE INHIBITORS MERCK & CO INC (US) 2007-10-31 EP disclosed
US-5366984-A Fungicides, insecticides BASF AKTIENGESELLSCHAFT (DE) 1994-11-22 US disclosed
US-5294628-A Fungicides, insecticides, pesticides BASF AKTIENGESELLSCHAFT (DE) 1994-03-15 US disclosed
EP-0378755-B1 Heterocyclically substituted alpha-aryl acryl acid methyl esters and their use BASF AG (DE) 1993-12-29 EP disclosed
US-5250553-A Fungicides; pesticides BASF AKTIENGESELLSCHAFT (DE) 1993-10-05 US disclosed
US-5166216-A Fungicides, pesticides, insecticides BASF AKTIENGESELLSCHAFT (DE) 1992-11-24 US disclosed
EP-0378755-A1 Heterocyclically substituted alpha-aryl acryl acid methyl esters and their use BASF Aktiengesellschaft (DE) 1990-07-25 EP disclosed