SCHEMBL7016863

SCHEMBL7016863

Cc1ccc(-n2ccc(C=O)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.50
MGLL Q99685 1/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39
TUBB3 Q13509 1/20 0.39
TUBB2A Q13885 1/20 0.39
TUBB8 Q3ZCM7 1/20 0.39
TUBA3E Q6PEY2 1/20 0.39
TUBA1A Q71U36 1/20 0.39
TUBA1C Q9BQE3 1/20 0.39
TUBB6 Q9BUF5 1/20 0.39
TUBB2B Q9BVA1 1/20 0.39
TUBB1 Q9H4B7 1/20 0.39
ALDH1A1 P00352 7/20 0.39
F2 P00734 1/20 0.38
ELANE P08246 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6052596 0.81 MGLL (0.39) MGLLTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL9309316 0.81 HSD17B10 (0.50) MGLLTUBB4ATUBBTUBA3CTUBA1B
SCHEMBL5126021 0.81 FAAH (0.39) MGLLALDH1A1GRIA1GRIA2GRIA3
SCHEMBL3095401 0.81 FAAH (0.39) MGLLALDH1A1GRIA1GRIA2GRIA3
SCHEMBL5116483 0.80 ALDH1A1 (0.55) CYP2A6MGLLTUBB4ATUBBTUBA3C
SCHEMBL1680730 0.80 COMT (0.48) CYP2A6MGLLTUBB4ATUBBTUBA3C
SCHEMBL8506107 0.79 PTGS2 (0.40)
SCHEMBL6630210 0.78 MEN1 (0.43) CYP2A6MGLLALDH1A1GRIA1GRIA2
SCHEMBL14395511 0.77 BCHE (0.39) ALDH1A1GRIA1GRIA2GRIA3GRIA4
SCHEMBL5129468 0.77 HDAC2 (0.37) CYP2A6ALDH1A1ELANEGRIA1GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1327631-A2 Fused heterocyclic compounds, their production and use as angiotensin II antagonists Takeda Chemical Industries, Ltd. (JP) 2003-07-16 EP disclosed
EP-0518033-B1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-07-02 EP disclosed
US-5484937-A ANGIOTENSIN ANTAGONISTS G.D. SEARLE & CO. (US) 1996-01-16 US disclosed
US-5389641-A Fused heterocyclic compounds, having angiotensin II antagonistic activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
US-5175180-A Antagonist, antagonism G. D. SEARLE & CO. (US) 1992-12-29 US disclosed
EP-0518033-A1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-12-16 EP disclosed
WO-1992011255-A1 N-SUBSTITUTED N-(α-TRIAZOLYL-TOLUYL)PYRROLE COMPOUNDS FOR TREATMENT OF CIRCULATORY DISORDERS G.D. SEARLE & CO. (US) 1992-07-09 WO disclosed