SCHEMBL9309824

SCHEMBL9309824

Cc1nc(Cl)c(Cc2ccc(-c3ccccc3C#N)cc2)c(C2CC2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.40
CNR2 P34972 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PRKAG1 P54619 3/20 0.38
PRKAA1 Q13131 3/20 0.38
PRKAB1 Q9Y478 3/20 0.38
ESR2 Q92731 1/20 0.37
ACHE P22303 2/20 0.36
FFAR1 O14842 1/20 0.35
AKR1B1 P15121 1/20 0.35
OXTR P30559 1/20 0.35
AVPR1A P37288 1/20 0.35
AKT1 P31749 2/20 0.35
AKT2 P31751 1/20 0.35
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
DPP4 P27487 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9309751 0.88 ESR2 (0.42) PPARGCNR2PRKAG1PRKAA1PRKAB1
SCHEMBL9309094 0.85 PPARG (0.36) PPARGCNR2CYP1A2CYP2C9CYP2C19
SCHEMBL1889453 0.81 KDM4E (0.41) PPARGCNR2CYP1A2CYP2C9CYP2C19
SCHEMBL9308998 0.80 KDM4E (0.37) PPARGCNR2CYP2C9CYP2C19PRKAG1
SCHEMBL1894428 0.79 PPARG (0.50) PPARGACHE
SCHEMBL1890638 0.78 CCR2 (0.39) PPARGCNR2CYP2C9CYP2C19ACHE
SCHEMBL9309290 0.77 PPARG (0.46) PPARGACHE
SCHEMBL9311500 0.76 AGTR1 (0.49) CYP2C9CYP2C19DPP4
SCHEMBL9309001 0.75 CNR1 (0.41) PPARGCNR2CYP2C9CYP2C19AKT1
SCHEMBL9311340 0.72 PPARG (0.49) PPARGESR2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5358950-A Useful in treatment of cardiovascular diseases LABORATOIRES UPSA (FR) 1994-10-25 US disclosed