SCHEMBL931100

SCHEMBL931100

COc1c(C)ccc(Br)c1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
NQO2 P16083 3/20 0.34
ALDH1A1 P00352 8/20 0.33
MAPT P10636 5/20 0.33
MEN1 O00255 4/20 0.33
HPGD P15428 4/20 0.33
KMT2A Q03164 4/20 0.33
APAF1 O14727 1/20 0.33
GAA P10253 3/20 0.32
PKM P14618 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.31
MPI P34949 1/20 0.31
KDM4E B2RXH2 2/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TUBB1 Q9H4B7 3/20 0.31
MGAM O43451 1/20 0.31
SI P14410 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26318648 0.83 NQO2 (0.38) CA2CA4NQO2ALDH1A1MAPT
SCHEMBL14405259 0.81 ALDH1A1 (0.36) ALDH1A1MAPTMEN1KMT2AGAA
SCHEMBL1223611 0.80 ALDH1A1 (0.44) CA2CA4NQO2ALDH1A1MAPT
SCHEMBL4922559 0.79 CA2 (0.44) CA2CA4NQO2ALDH1A1MAPT
SCHEMBL7484583 0.77 CA2 (0.48) CA2CA4NQO2ALDH1A1MAPT
SCHEMBL287639 0.77 CA2 (0.38) CA2CA4NQO2ALDH1A1MAPT
SCHEMBL21567219 0.77 L3MBTL1 (0.41) ALDH1A1MAPTMEN1HPGDKMT2A
SCHEMBL3836832 0.77 ALOX5AP (0.35) CA2CA4NQO2ALDH1A1MAPT
SCHEMBL30407777 0.77 ALOX5AP (0.38) CA2CA4NQO2ALDH1A1MAPT
SCHEMBL19629222 0.74 HTR2A (0.35) ALDH1A1MAPTGAAKDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002409-A1 5H-PYRROLO[3,4-£>]PYRAZIN-7-AMINE DERIVATIVES INHIBITORS OF BETA-SECRETASE ASTRAZENECA AB (SE) 2011-01-06 WO disclosed