SCHEMBL9311925

SCHEMBL9311925

COc1ccc(N2CCN(c3ccc(Cl)nn3)CC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
LMNA P02545 1/20 0.58
CYP1A2 P05177 1/20 0.54
BPTF Q12830 1/20 0.51
MAPT P10636 5/20 0.51
RAB9A P51151 3/20 0.51
KMT2A Q03164 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.50
L3MBTL1 Q9Y468 3/20 0.50
NPC1 O15118 2/20 0.50
MEN1 O00255 2/20 0.50
HTR3E A5X5Y0 1/20 0.49
HTR3B O95264 1/20 0.49
ADRB1 P08588 1/20 0.49
HTR3A P46098 1/20 0.49
HTR3D Q70Z44 1/20 0.49
HTR3C Q8WXA8 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
DRD2 P14416 1/20 0.48
DPP4 P27487 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9212665 0.79 DRD2 (0.52) ALDH1A1LMNAMAPTSIGMAR1DRD2
SCHEMBL29656856 0.78 HTR3E (0.73) ALDH1A1LMNAMAPTRAB9AKMT2A
SCHEMBL28599511 0.78 HTR3E (0.73) ALDH1A1LMNAMAPTRAB9AKMT2A
SCHEMBL28432321 0.77 MAPT (0.64) ALDH1A1LMNAMAPTRAB9AKMT2A
SCHEMBL3023133 0.77 MAPT (0.58) ALDH1A1CYP1A2MAPTRAB9AKMT2A
SCHEMBL9311771 0.76 MAPT (0.59) ALDH1A1LMNAMAPTRAB9AKMT2A
SCHEMBL257823 0.75 CYP1A2 (0.67) ALDH1A1LMNACYP1A2BPTFMAPT
SCHEMBL9311935 0.74 LMNA (1.00) ALDH1A1LMNACYP1A2MAPTRAB9A
SCHEMBL15887431 0.73 HTR3E (0.61) ALDH1A1LMNAMAPTRAB9AKMT2A
SCHEMBL13390484 0.73 HTR3E (0.61) ALDH1A1LMNAMAPTRAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5292738-A Anti-virally active pyridazinamines JANSSEN PHARMACEUTICA N.V. (BE) 1994-03-08 US disclosed
US-5157035-A Viricides JANSSEN PHARMACEUTICA N. V. (BE) 1992-10-20 US disclosed
US-5001125-A Anti-virally active pyridazinamines JANSSEN PHARMACEUTICA N.V. (BE) 1991-03-19 US disclosed
EP-0156433-B1 ANTI-VIRALLY ACTIVE PYRIDAZINAMINES JANSSEN PHARMACEUTICA N.V. (BE) 1991-02-27 EP disclosed
EP-0156433-A2 Anti-virally active pyridazinamines JANSSEN PHARMACEUTICA N.V. (BE) 1985-10-02 EP disclosed