SCHEMBL9312484

SCHEMBL9312484

COc1cccc(/C=C/C(=O)Nc2ccc3c(c2)NC(=O)CC3(C)C)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
MAPT P10636 3/20 0.56
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
NFKB1 P19838 1/20 0.56
NFKB2 Q00653 1/20 0.56
RELA Q04206 1/20 0.56
MMP1 P03956 6/20 0.55
MMP2 P08253 6/20 0.55
MMP9 P14780 6/20 0.55
LMNA P02545 1/20 0.53
TRPV1 Q8NER1 4/20 0.52
ACHE P22303 1/20 0.50
HDAC6 Q9UBN7 2/20 0.49
TP53 P04637 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9312489 1.00 ALDH1A1 (0.59) ALDH1A1SMN1; SMN2MAPTKMT2AMEN1
SCHEMBL9313174 0.89 MAPT (0.55) ALDH1A1SMN1; SMN2MAPTKMT2AMEN1
SCHEMBL9313168 0.89 MAPT (0.55) ALDH1A1SMN1; SMN2MAPTKMT2AMEN1
SCHEMBL9313383 0.87 MAPT (0.55) ALDH1A1SMN1; SMN2MAPTKMT2AMEN1
SCHEMBL9313377 0.87 MAPT (0.55) ALDH1A1SMN1; SMN2MAPTKMT2AMEN1
SCHEMBL10587887 0.85 SMN1; SMN2 (0.62) ALDH1A1SMN1; SMN2MAPTKMT2AMEN1
SCHEMBL10587883 0.85 SMN1; SMN2 (0.62) ALDH1A1SMN1; SMN2MAPTKMT2AMEN1
SCHEMBL9312470 0.82 TRPV1 (0.56) MMP1MMP2MMP9TRPV1HDAC6
SCHEMBL9312463 0.82 TRPV1 (0.56) MMP1MMP2MMP9TRPV1HDAC6
SCHEMBL9313855 0.82 MAPT (0.59) ALDH1A1SMN1; SMN2MAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5373019-A Pharmaceutical lactam compositions for inhibition of erythrocyte and thrombocyte aggregation BOEHRINGER MANNHEIM GMBH (DE) 1994-12-13 US disclosed
US-4985448-A Ureidoindoles, pharmaceutical compositions and methods for erythrocyte and thrombocyte aggregation inhibition BOEHRINGER MANNHEIM GMBH (DE) 1991-01-15 US disclosed