SCHEMBL10587883

SCHEMBL10587883

COc1cccc(C=CC(=O)Nc2ccc3c(c2)NC(=O)C3(C)C)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.62
ALDH1A1 P00352 3/20 0.62
MMP1 P03956 6/20 0.58
MMP2 P08253 6/20 0.58
MMP9 P14780 6/20 0.58
MAPT P10636 4/20 0.57
KMT2A Q03164 4/20 0.57
MEN1 O00255 3/20 0.57
NPC1 O15118 3/20 0.57
RAB9A P51151 3/20 0.57
NFKB1 P19838 1/20 0.57
NFKB2 Q00653 1/20 0.57
RELA Q04206 1/20 0.57
LMNA P02545 2/20 0.56
TRPV1 Q8NER1 3/20 0.55
ACHE P22303 1/20 0.52
TP53 P04637 2/20 0.52
HDAC6 Q9UBN7 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10587887 1.00 SMN1; SMN2 (0.62) SMN1; SMN2ALDH1A1MMP1MMP2MMP9
SCHEMBL10588017 0.89 MAPT (0.58) SMN1; SMN2ALDH1A1MMP1MMP2MMP9
SCHEMBL10588022 0.89 MAPT (0.58) SMN1; SMN2ALDH1A1MMP1MMP2MMP9
SCHEMBL10478111 0.86 MAPT (0.58) SMN1; SMN2ALDH1A1MMP1MMP2MMP9
SCHEMBL9312217 0.86 MAPT (0.58) SMN1; SMN2ALDH1A1MMP1MMP2MMP9
SCHEMBL9312484 0.85 ALDH1A1 (0.59) SMN1; SMN2ALDH1A1MMP1MMP2MMP9
SCHEMBL9312489 0.85 ALDH1A1 (0.59) SMN1; SMN2ALDH1A1MMP1MMP2MMP9
SCHEMBL9312296 0.81 MMP1 (0.57) ALDH1A1MMP1MMP2MMP9MAPT
SCHEMBL9312300 0.81 MMP1 (0.57) ALDH1A1MMP1MMP2MMP9MAPT
SCHEMBL10585350 0.77 MAOB (0.54) ALDH1A1MAPTTRPV1ACHEKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0327986-A2 Medicaments containing lactams, substituted lactams and process for their preparation Roche Diagnostics GmbH (DE) 1989-08-16 EP disclosed